# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5279363 | 58 | INH | 0 | ALA5226244 | Active | % | Homo sapiens | ||||
2. | ALA5279363 | 58 | IC50 | > | 10 | uM | ALA5226243 | nM | Homo sapiens | |||
3. | ALA5279363 | 58 | IC50 | > | 10 | uM | ALA5226242 | nM | Homo sapiens | |||
4. | ALA5279363 | 58 | IC50 | > | 10 | uM | ALA5226241 | nM | Homo sapiens | |||
5. | ALA5279363 | 58 | IC50 | > | 10 | uM | ALA5226240 | nM | Homo sapiens | |||
6. | ALA5279363 | 58 | IC50 | > | 10 | uM | ALA5226239 | nM | Homo sapiens | |||
7. | ALA5279363 | 58 | IC50 | > | 10 | uM | ALA5226238 | nM | Homo sapiens | |||
8. | ALA5279363 | 58 | FC | = | 100 | ALA5226237 | Homo sapiens | |||||
9. | ALA5279363 | 58 | FC | = | 100 | ALA5226236 | Homo sapiens | |||||
10. | ALA5279363 | 58 | FC | = | 100 | ALA5226235 | Homo sapiens | |||||
11. | ALA5279363 | 58 | FC | = | 100 | ALA5226234 | Homo sapiens | |||||
12. | ALA5279363 | 58 | FC | = | 100 | ALA5226233 | Homo sapiens | |||||
13. | ALA5279363 | 58 | FC | = | 100 | ALA5226232 | Homo sapiens | |||||
14. | ALA5279363 | 58 | F | = | 47 | % | ALA5226231 | % | ||||
15. | ALA5279363 | 58 | F | = | 36 | % | ALA5226230 | % | ||||
16. | ALA5279363 | 58 | Cmax | = | 2270 | nM | ALA5226229 | nM | ||||
17. | ALA5279363 | 58 | Cmax | = | 1310 | nM | ALA5226228 | nM | ||||
18. | ALA5279363 | 58 | AUC | = | 4290 | hr.ng/ml | ALA5226227 | ng.hr.mL-1 | ||||
19. | ALA5279363 | 58 | AUC | = | 1338 | hr.ng/ml | ALA5226226 | ng.hr.mL-1 | ||||
20. | ALA5279363 | 58 | t1/2 | = | 6.1 | hr | ALA5226225 | hr |