# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5279688 | 25c | F | = | 9.14 | % | ALA5241996 | % | ||||
2. | ALA5279688 | 25c | t1/2 | = | 1.11 | hr | ALA5241995 | hr | ||||
3. | ALA5279688 | 25c | AUC | = | 1598.83 | ug/L.hr | ALA5241994 | ng.hr.mL-1 | ||||
4. | ALA5279688 | 25c | AUCt | = | 1591.06 | ug/L.hr | ALA5241993 | ng.hr.mL-1 | ||||
5. | ALA5279688 | 25c | Tmax | = | 3.33 | hr | ALA5241992 | hr | ||||
6. | ALA5279688 | 25c | Cmax | = | 372.9 | ug ml-1 | ALA5241991 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
7. | ALA5279688 | 25c | Vz | = | 1.74 | L/Kg | ALA5241990 | L.kg-1 | ||||
8. | ALA5279688 | 25c | CL | = | 1.48 | L/hr.Kg | ALA5241989 | mL.min-1.kg-1 | ||||
9. | ALA5279688 | 25c | t1/2 | = | 0.82 | hr | ALA5241988 | hr | ||||
10. | ALA5279688 | 25c | AUC | = | 3484.88 | ug/L.hr | ALA5241987 | ng.hr.mL-1 | ||||
11. | ALA5279688 | 25c | AUCt | = | 3481.96 | ug/L.hr | ALA5241986 | ng.hr.mL-1 | ||||
12. | ALA5279688 | 25c | Tmax | = | 0.08 | hr | ALA5241985 | hr | ||||
13. | ALA5279688 | 25c | Cmax | = | 4973.96 | ug ml-1 | ALA5241984 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
14. | ALA5279688 | 25c | t1/2 | = | 15.61 | min | ALA5241983 | hr | ||||
15. | ALA5279688 | 25c | t1/2 | = | 27.11 | min | ALA5241982 | hr | ||||
16. | ALA5279688 | 25c | IC50 | = | 14.36 | uM | ALA5241969 | 4.84 | nM | Homo sapiens | ||
17. | ALA5279688 | 25c | IC50 | = | 5.76 | uM | ALA5241968 | 5.24 | nM | Homo sapiens | ||
18. | ALA5279688 | 25c | IC50 | = | 9.22 | uM | ALA5241967 | 5.04 | nM | Homo sapiens | ||
19. | ALA5279688 | 25c | deltaTm | = | 11.8 | degrees C | ALA5241966 | degrees C | Homo sapiens | |||
20. | ALA5279688 | 25c | IC50 | > | 20 | uM | ALA5241965 | nM | Homo sapiens |