| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5279890 | (3R,4S)-10a | Emax | = | 216.5 | % | ALA5227869 | % | Homo sapiens | |||
| 2. | ALA5279890 | (3R,4S)-10a | EC50 | = | 1032 | nM | ALA5227868 | 5.99 | nM | Homo sapiens | ||
| 3. | ALA5279890 | (3R,4S)-10a | Emax | = | 215.8 | % | ALA5227867 | % | Homo sapiens | |||
| 4. | ALA5279890 | (3R,4S)-10a | EC50 | = | 133.6 | nM | ALA5227866 | 6.87 | nM | Homo sapiens | ||
| 5. | ALA5279890 | (3R,4S)-10a | Emax | = | 238.5 | % | ALA5227865 | % | Homo sapiens | |||
| 6. | ALA5279890 | (3R,4S)-10a | EC50 | = | 18.6 | nM | ALA5227864 | 7.73 | nM | Homo sapiens | ||
| 7. | ALA5279890 | (3R,4S)-10a | Selectivity ratio | = | 70.5 | ALA5227862 | ||||||
| 8. | ALA5279890 | (3R,4S)-10a | Selectivity ratio | = | 99.1 | ALA5227861 | ||||||
| 9. | ALA5279890 | (3R,4S)-10a | Ki | = | 126.9 | nM | ALA5227857 | 6.90 | nM | Homo sapiens | ||
| 10. | ALA5279890 | (3R,4S)-10a | Ki | = | 178.3 | nM | ALA5227856 | 6.75 | nM | Homo sapiens | ||
| 11. | ALA5279890 | (3R,4S)-10a | Ki | = | 1.8 | nM | ALA5227855 | 8.74 | nM | Mus musculus | ||
| 12. | ALA5279890 | (3R,4S)-10a | ED50 | = | 0.4 | ug | ALA5227853 | ug | Mus musculus |
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