| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5280464 | 26 | INH | <= | 100 | % | ALA5239271 | % | Homo sapiens | |||
| 2. | ALA5280464 | 26 | INH | = | 13 | % | ALA5239270 | % | Mus musculus | |||
| 3. | ALA5280464 | 26 | INH | = | 30 | % | ALA5239268 | % | Sus scrofa | |||
| 4. | ALA5280464 | 26 | IC50 | = | 41 | uM | ALA5239266 | 4.39 | nM | Homo sapiens | ||
| 5. | ALA5280464 | 26 | Activity | = | 80.5 | % | ALA5239265 | % | ||||
| 6. | ALA5280464 | 26 | PPB | = | 68.7 | % | ALA5239264 | % | ||||
| 7. | ALA5280464 | 26 | CL | = | 16.5 | microL/min/mg | ALA5239263 | mL.min-1.g-1 | ||||
| 8. | ALA5280464 | 26 | t1/2 | > | 40 | min | ALA5239262 | hr | ||||
| 9. | ALA5280464 | 26 | t1/2 | > | 6 | hr | ALA5239261 | hr | ||||
| 10. | ALA5280464 | 26 | logD | = | 0.243 | ALA5239260 | ||||||
| 11. | ALA5280464 | 26 | solubility | >= | 200 | uM | ALA5239259 | nM | ||||
| 12. | ALA5280464 | 26 | MIC | = | 0.06 | ug ml-1 | ALA5239236 | ug.mL-1 | Pseudomonas aeruginosa | |||
| 13. | ALA5280464 | 26 | MIC | = | 16 | ug ml-1 | ALA5239235 | ug.mL-1 | Pseudomonas aeruginosa | |||
| 14. | ALA5280464 | 26 | MIC | = | 0.03 | ug ml-1 | ALA5239234 | ug.mL-1 | Klebsiella pneumoniae | |||
| 15. | ALA5280464 | 26 | MIC | = | 0.06 | ug ml-1 | ALA5239233 | ug.mL-1 | Klebsiella pneumoniae | |||
| 16. | ALA5280464 | 26 | Activity | 0 | ALA5239232 | Not Active | ||||||
| 17. | ALA5280464 | 26 | Activity | 0 | ALA5239231 | Not Active | ||||||
| 18. | ALA5280464 | 26 | deltaH | = | 6 | kcal/mol | ALA5239225 | kcal/mol | ||||
| 19. | ALA5280464 | 26 | Kd | = | 10 | nM | ALA5239224 | 8.00 | nM | |||
| 20. | ALA5280464 | 26 | INH | 0 | ALA5239221 | Active | % |
The page will load shortly, Thanks for your patience!