# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5280568 | (R)-30; BRD9500 | Activity | 0 | ALA5264801 | Active | Homo sapiens | |||||
2. | ALA5280568 | (R)-30; BRD9500 | Ratio IC50/EC50 | = | 2.4 | ALA5264800 | ||||||
3. | ALA5280568 | (R)-30; BRD9500 | Ratio IC50/EC50 | = | 2.4 | ALA5264799 | ||||||
4. | ALA5280568 | (R)-30; BRD9500 | IC50 | = | 10 | nM | ALA5264797 | 8.00 | nM | Homo sapiens | ||
5. | ALA5280568 | (R)-30; BRD9500 | Activity | 0 | ALA5264796 | Not Active | Homo sapiens | |||||
6. | ALA5280568 | (R)-30; BRD9500 | EC50 | = | 1.6 | nM | ALA5264795 | 8.80 | nM | Homo sapiens | ||
7. | ALA5280568 | (R)-30; BRD9500 | Activity | 0 | ALA5264794 | Not Active | Homo sapiens | |||||
8. | ALA5280568 | (R)-30; BRD9500 | Activity | 0 | ALA5264792 | Not Active | Homo sapiens | |||||
9. | ALA5280568 | (R)-30; BRD9500 | INH | 0 | ALA5264791 | Not Active | % | Homo sapiens | ||||
10. | ALA5280568 | (R)-30; BRD9500 | INH | 0 | ALA5264790 | Not Active | % | |||||
11. | ALA5280568 | (R)-30; BRD9500 | INH | 0 | ALA5264789 | Not Active | % | Homo sapiens | ||||
12. | ALA5280568 | (R)-30; BRD9500 | INH | 0 | ALA5264788 | Not Active | % | Homo sapiens | ||||
13. | ALA5280568 | (R)-30; BRD9500 | INH | 0 | ALA5264787 | Not Active | % | Homo sapiens | ||||
14. | ALA5280568 | (R)-30; BRD9500 | INH | 0 | ALA5264786 | Not Active | % | Homo sapiens | ||||
15. | ALA5280568 | (R)-30; BRD9500 | INH | 0 | ALA5264785 | Not Active | % | Homo sapiens | ||||
16. | ALA5280568 | (R)-30; BRD9500 | INH | 0 | ALA5264784 | Not Active | % | Homo sapiens | ||||
17. | ALA5280568 | (R)-30; BRD9500 | INH | 0 | ALA5264783 | Not Active | % | Homo sapiens | ||||
18. | ALA5280568 | (R)-30; BRD9500 | INH | 0 | ALA5264782 | Not Active | % | Homo sapiens | ||||
19. | ALA5280568 | (R)-30; BRD9500 | EC50 | = | 1.3 | nM | ALA5264781 | 8.89 | nM | Homo sapiens | ||
20. | ALA5280568 | (R)-30; BRD9500 | solubility | = | 1 | mM | ALA5264780 | nM |