# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5283388 | 6 | Ratio | = | 0.058 | ALA5239613 | ||||||
2. | ALA5283388 | 6 | Ratio | = | 0.074 | ALA5239612 | ||||||
3. | ALA5283388 | 6 | Ratio | = | 0.139 | ALA5239611 | ||||||
4. | ALA5283388 | 6 | Ratio | = | 0.209 | ALA5239610 | ||||||
5. | ALA5283388 | 6 | Ct | = | 15.6 | nM | ALA5239609 | nM | ||||
6. | ALA5283388 | 6 | Ct | = | 53.1 | nM | ALA5239608 | nM | ||||
7. | ALA5283388 | 6 | Ct | = | 37.1 | nM | ALA5239607 | nM | ||||
8. | ALA5283388 | 6 | Ct | = | 150 | nM | ALA5239606 | nM | ||||
9. | ALA5283388 | 6 | Cp | = | 267 | nM | ALA5239605 | nM | ||||
10. | ALA5283388 | 6 | Cp | = | 717 | nM | ALA5239604 | nM | ||||
11. | ALA5283388 | 6 | Fu | = | 0.081 | % | ALA5239603 | |||||
12. | ALA5283388 | 6 | Stability | = | 70.7 | ml/min.kg | ALA5239602 | ml/min.kg | ||||
13. | ALA5283388 | 6 | permeability | > | 50 | 10^-6 cm/s | ALA5239601 | 10^-6 cm/s | ||||
14. | ALA5283388 | 6 | solubility | = | 28.3 | uM | ALA5239600 | nM | ||||
15. | ALA5283388 | 6 | solubility | = | 0.66 | uM | ALA5239599 | nM | ||||
16. | ALA5283388 | 6 | TdeltaS | = | 6 | kcal/mol | ALA5239598 | kcal/mol | Homo sapiens | |||
17. | ALA5283388 | 6 | deltaH | = | -16.68 | kcal/mol | ALA5239597 | kcal/mol | Homo sapiens | |||
18. | ALA5283388 | 6 | deltaG | = | -10.67 | kcal/mol | ALA5239596 | kcal/mol | Homo sapiens | |||
19. | ALA5283388 | 6 | Kd | = | 16 | nM | ALA5239595 | 7.80 | nM | Homo sapiens | ||
20. | ALA5283388 | 6 | IC5 | = | 3.7 | uM | ALA5239594 | uM | Homo sapiens |