| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5283820 | 17c | BPR | = | 7.3 | ALA5223858 | ||||||
| 2. | ALA5283820 | 17c | CL | = | 124 | ml/min.kg | ALA5223857 | mL.min-1.kg-1 | ||||
| 3. | ALA5283820 | 17c | Vdss | = | 19.5 | L/Kg | ALA5223856 | L.kg-1 | ||||
| 4. | ALA5283820 | 17c | beta t1/2 | = | 1.8 | hr | ALA5223855 | hr | ||||
| 5. | ALA5283820 | 17c | AUC | = | 31 | ng.hr/ml | ALA5223854 | ng.hr.mL-1 | ||||
| 6. | ALA5283820 | 17c | Cmax | = | 12 | ng/ml | ALA5223853 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 7. | ALA5283820 | 17c | F | = | 7 | % | ALA5223852 | % | ||||
| 8. | ALA5283820 | 17c | Drug metabolism | = | 44.4 | % | ALA5223846 | % | ||||
| 9. | ALA5283820 | 17c | Drug metabolism | = | 73 | % | ALA5223845 | % | ||||
| 10. | ALA5283820 | 17c | Emax | = | 53 | % | ALA5223844 | % | Homo sapiens | |||
| 11. | ALA5283820 | 17c | EC50 | = | 8.6 | nM | ALA5223843 | 8.07 | nM | Homo sapiens |
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