| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5284082 | 2g | Ratio | = | 0.65 | ALA5252406 | ||||||
| 2. | ALA5284082 | 2g | F | 0 | ALA5252405 | Not Determined | % | |||||
| 3. | ALA5284082 | 2g | Vdss | 0 | ALA5252404 | Not Determined | ||||||
| 4. | ALA5284082 | 2g | CL | 0 | ALA5252403 | Not Determined | ||||||
| 5. | ALA5284082 | 2g | t1/2 | = | 13.5 | hr | ALA5252402 | hr | ||||
| 6. | ALA5284082 | 2g | AUC | = | 23.6 | uM.hr | ALA5252401 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 7. | ALA5284082 | 2g | Tmax | = | 6 | hr | ALA5252400 | hr | ||||
| 8. | ALA5284082 | 2g | Cmax | = | 1.4 | uM | ALA5252399 | nM | ||||
| 9. | ALA5284082 | 2g | Activity | 0 | ALA5252398 | Not Active | Mus musculus | |||||
| 10. | ALA5284082 | 2g | Activity | 0 | ALA5252396 | Active | Mus musculus | |||||
| 11. | ALA5284082 | 2g | Efficacy | = | 64 | % | ALA5252395 | % | Mus musculus | |||
| 12. | ALA5284082 | 2g | Fu | = | 0.7 | % | ALA5252394 | |||||
| 13. | ALA5284082 | 2g | Therm_solubility | = | 25 | uM | ALA5252393 | nM | ||||
| 14. | ALA5284082 | 2g | logD | = | 0.6 | ALA5252392 | ||||||
| 15. | ALA5284082 | 2g | INH | = | -2.9 | % | ALA5252391 | % | Homo sapiens | |||
| 16. | ALA5284082 | 2g | Ratio IC50 | = | 30 | ALA5252389 | ||||||
| 17. | ALA5284082 | 2g | IC50 | = | 32 | uM | ALA5252388 | 4.50 | nM | Homo sapiens | ||
| 18. | ALA5284082 | 2g | IC50 | = | 1.2 | uM | ALA5252387 | 5.92 | nM | Homo sapiens | ||
| 19. | ALA5284082 | 2g | IC50 | = | 0.015 | uM | ALA5252385 | 7.82 | nM | Mus musculus | ||
| 20. | ALA5284082 | 2g | IC50 | = | 0.04 | uM | ALA5252384 | 7.40 | nM | Homo sapiens |
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