| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5284303 | R-26j; RK-0133114 | INH | 0 | ALA5251553 | Not Active | % | Mus musculus | ||||
| 2. | ALA5284303 | R-26j; RK-0133114 | Cp | = | 18.9 | uM | ALA5251552 | uM | ||||
| 3. | ALA5284303 | R-26j; RK-0133114 | Cp | = | 9.6 | uM | ALA5251551 | uM | ||||
| 4. | ALA5284303 | R-26j; RK-0133114 | Ct | = | 46.9 | uM | ALA5251550 | uM | ||||
| 5. | ALA5284303 | R-26j; RK-0133114 | Ct | = | 23.5 | uM | ALA5251549 | uM | ||||
| 6. | ALA5284303 | R-26j; RK-0133114 | Activity | 0 | ALA5251548 | Active | Mus musculus | |||||
| 7. | ALA5284303 | R-26j; RK-0133114 | Activity | 0 | ALA5251547 | Non-Toxic | ||||||
| 8. | ALA5284303 | R-26j; RK-0133114 | Activity | 0 | ALA5251546 | Active | ||||||
| 9. | ALA5284303 | R-26j; RK-0133114 | t1/2 | = | 1.4 | hr | ALA5251545 | hr | ||||
| 10. | ALA5284303 | R-26j; RK-0133114 | Tmax | = | 4 | hr | ALA5251544 | hr | ||||
| 11. | ALA5284303 | R-26j; RK-0133114 | AUC | = | 418 | umol/l.hr | ALA5251543 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 12. | ALA5284303 | R-26j; RK-0133114 | Cmax | = | 42.4 | umol/L | ALA5251542 | nM | ||||
| 13. | ALA5284303 | R-26j; RK-0133114 | Activity | 0 | ALA5251541 | Not Active | ||||||
| 14. | ALA5284303 | R-26j; RK-0133114 | GI50 | = | 2370 | nM | ALA5251539 | nM | Homo sapiens | |||
| 15. | ALA5284303 | R-26j; RK-0133114 | IC50 | = | 3700 | nM | ALA5251534 | 5.43 | nM | Homo sapiens | ||
| 16. | ALA5284303 | R-26j; RK-0133114 | IC50 | = | 53 | nM | ALA5251533 | 7.28 | nM | Homo sapiens | ||
| 17. | ALA5284303 | R-26j; RK-0133114 | IC50 | = | 27 | nM | ALA5251532 | 7.57 | nM | Homo sapiens |
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