| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5285249 | 5 | K(p,uu,brain) | = | 0.2 | ALA5256789 | ||||||
| 2. | ALA5285249 | 5 | BPR | = | 0.22 | ALA5256788 | ||||||
| 3. | ALA5285249 | 5 | AUC | = | 529 | ng.hr/ml | ALA5256787 | ng.hr.mL-1 | ||||
| 4. | ALA5285249 | 5 | t1/2 | = | 1.54 | hr | ALA5256786 | hr | ||||
| 5. | ALA5285249 | 5 | Tmax | = | 1 | hr | ALA5256785 | hr | ||||
| 6. | ALA5285249 | 5 | Cmax | = | 0.6 | uM | ALA5256784 | nM | ||||
| 7. | ALA5285249 | 5 | F | = | 19 | % | ALA5256783 | % | ||||
| 8. | ALA5285249 | 5 | Vdss | = | 0.94 | L/Kg | ALA5256782 | L.kg-1 | ||||
| 9. | ALA5285249 | 5 | CL | = | 18 | ml/min.kg | ALA5256781 | mL.min-1.kg-1 | ||||
| 10. | ALA5285249 | 5 | Ratio | = | 0.9 | ALA5256780 | ||||||
| 11. | ALA5285249 | 5 | Papp | = | 119 | nm/s | ALA5256779 | nm/s | ||||
| 12. | ALA5285249 | 5 | Fu | = | 0.247 | ALA5256778 | ||||||
| 13. | ALA5285249 | 5 | Fu | = | 0.279 | ALA5256777 | ||||||
| 14. | ALA5285249 | 5 | CLH | = | 27 | ml/min.kg | ALA5256776 | mL.min-1.kg-1 | ||||
| 15. | ALA5285249 | 5 | CLH | < | 14 | ml/min.kg | ALA5256775 | mL.min-1.kg-1 | ||||
| 16. | ALA5285249 | 5 | CLH | = | 0.01 | microL/min/mg | ALA5256774 | mL.min-1.g-1 | ||||
| 17. | ALA5285249 | 5 | CLH | = | 0.01 | microL/min/mg | ALA5256773 | mL.min-1.g-1 | ||||
| 18. | ALA5285249 | 5 | Emax | = | 100 | % | ALA5256772 | % | Homo sapiens | |||
| 19. | ALA5285249 | 5 | EC50 | = | 6 | nM | ALA5256771 | 8.22 | nM | Homo sapiens |
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