# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5285607 | 16; OFH5503 | Activity | 0 | ALA5239865 | Not Active | Homo sapiens | |||||
2. | ALA5285607 | 16; OFH5503 | Activity | 0 | ALA5239864 | Not Active | Homo sapiens | |||||
3. | ALA5285607 | 16; OFH5503 | Activity | 0 | ALA5239863 | Active | Homo sapiens | |||||
4. | ALA5285607 | 16; OFH5503 | Activity | 0 | ALA5239862 | Active | Homo sapiens | |||||
5. | ALA5285607 | 16; OFH5503 | pKi | = | 9.88 | ALA5239861 | 9.88 | nM | Homo sapiens | |||
6. | ALA5285607 | 16; OFH5503 | Ki | = | 0.15 | nM | ALA5239861 | 9.82 | nM | Homo sapiens | ||
7. | ALA5285607 | 16; OFH5503 | pKi | = | 8.66 | ALA5239860 | 8.66 | nM | Homo sapiens | |||
8. | ALA5285607 | 16; OFH5503 | Ki | = | 2.3 | nM | ALA5239860 | 8.64 | nM | Homo sapiens | ||
9. | ALA5285607 | 16; OFH5503 | Activity | 0 | ALA5239859 | Non-Toxic | Cricetulus griseus | |||||
10. | ALA5285607 | 16; OFH5503 | Kdiss | = | 0.024 | /min | ALA5239858 | /min | Homo sapiens | |||
11. | ALA5285607 | 16; OFH5503 | ka | = | 0.37 | /min | ALA5239856 | /min | Homo sapiens | |||
12. | ALA5285607 | 16; OFH5503 | Kd | = | 7.3 | nM | ALA5239854 | 8.14 | nM | Homo sapiens | ||
13. | ALA5285607 | 16; OFH5503 | Kd | = | 8.3 | nM | ALA5239853 | 8.08 | nM | Homo sapiens | ||
14. | ALA5285607 | 16; OFH5503 | Kd | = | 24 | nM | ALA5239852 | 7.62 | nM | Homo sapiens | ||
15. | ALA5285607 | 16; OFH5503 | Kd | = | 23 | nM | ALA5239851 | 7.64 | nM | Homo sapiens | ||
16. | ALA5285607 | 16; OFH5503 | IC50 | = | 430 | nM | ALA5239848 | 6.37 | nM | Homo sapiens | ||
17. | ALA5285607 | 16; OFH5503 | IC50 | = | 130 | nM | ALA5239847 | 6.89 | nM | Homo sapiens | ||
18. | ALA5285607 | 16; OFH5503 | Selectivity ratio | = | 6.2 | ALA5239846 | ||||||
19. | ALA5285607 | 16; OFH5503 | Selectivity ratio | = | 1.2 | ALA5239845 | ||||||
20. | ALA5285607 | 16; OFH5503 | Selectivity ratio | = | 9.2 | ALA5239844 | Homo sapiens |