# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5287177 | 22 | Fu | = | 0.022 | ALA5224121 | ||||||
2. | ALA5287177 | 22 | AUC | = | 116 | uM.hr | ALA5224119 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
3. | ALA5287177 | 22 | Cmax | = | 22.6 | uM | ALA5224118 | nM | ||||
4. | ALA5287177 | 22 | Fu | = | 0.022 | ALA5224117 | ||||||
5. | ALA5287177 | 22 | Cp | = | 0.016 | uM | ALA5224116 | uM | ||||
6. | ALA5287177 | 22 | AUC | = | 25.7 | uM.hr | ALA5224115 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
7. | ALA5287177 | 22 | Cmax | = | 6.1 | uM | ALA5224114 | nM | ||||
8. | ALA5287177 | 22 | Kinetic_solubility | = | 209 | uM | ALA5224113 | nM | ||||
9. | ALA5287177 | 22 | Kinetic_solubility | = | 0 | uM | ALA5224112 | nM | ||||
10. | ALA5287177 | 22 | Kinetic_solubility | = | 500 | uM | ALA5224111 | nM | ||||
11. | ALA5287177 | 22 | IC50 | = | 0.077 | uM | ALA5224110 | 7.11 | nM | Mus musculus | ||
12. | ALA5287177 | 22 | permeability | < | 3 | nm/s | ALA5224109 | nm/s | ||||
13. | ALA5287177 | 22 | Time | >= | 12 | hr | ALA5224108 | hr | Homo sapiens | |||
14. | ALA5287177 | 22 | Activity | 0 | ALA5224106 | Not Active | Homo sapiens | |||||
15. | ALA5287177 | 22 | Drug uptake | = | 17.5 | uM | ALA5224105 | uM | ||||
16. | ALA5287177 | 22 | Cp | = | 5.7 | uM | ALA5224104 | uM | ||||
17. | ALA5287177 | 22 | Activity | 0 | ALA5224103 | Active | Homo sapiens | |||||
18. | ALA5287177 | 22 | Cp | = | 0.03 | uM | ALA5224102 | uM | ||||
19. | ALA5287177 | 22 | Fu | = | 0.022 | ALA5224101 | ||||||
20. | ALA5287177 | 22 | F | = | 35 | % | ALA5224100 | % |