| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5288241 | B2 | F | = | 64.2 | % | ALA5238312 | % | ||||
| 2. | ALA5288241 | B2 | Activity | 0 | ALA5238311 | Active | Mus musculus | |||||
| 3. | ALA5288241 | B2 | INH | 0 | ALA5238310 | Active | % | Mus musculus | ||||
| 4. | ALA5288241 | B2 | Activity | 0 | ALA5238309 | Non-Toxic | ||||||
| 5. | ALA5288241 | B2 | Activity | 0 | ALA5238308 | Non-Toxic | ||||||
| 6. | ALA5288241 | B2 | Activity | 0 | ALA5238307 | Active | Mus musculus | |||||
| 7. | ALA5288241 | B2 | Activity | 0 | ALA5238306 | Active | Mus musculus | |||||
| 8. | ALA5288241 | B2 | Activity | 0 | ALA5238305 | Active | Mus musculus | |||||
| 9. | ALA5288241 | B2 | INH | 0 | ALA5238304 | Dose-Dependent Effect | % | Mus musculus | ||||
| 10. | ALA5288241 | B2 | IC50 | = | 13 | uM | ALA5238303 | 4.89 | nM | Homo sapiens | ||
| 11. | ALA5288241 | B2 | INH | 0 | ALA5238302 | Dose-Dependent Effect | % | |||||
| 12. | ALA5288241 | B2 | MRT | = | 5 | hr | ALA5238301 | hr | ||||
| 13. | ALA5288241 | B2 | Cmax | = | 3806 | ng/ml | ALA5238300 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 14. | ALA5288241 | B2 | Tmax | = | 1 | hr | ALA5238299 | hr | ||||
| 15. | ALA5288241 | B2 | t1/2 | = | 3 | hr | ALA5238298 | hr | ||||
| 16. | ALA5288241 | B2 | AUC | = | 17411 | hr.ng/ml | ALA5238297 | ng.hr.mL-1 | ||||
| 17. | ALA5288241 | B2 | AUClast | = | 17280 | hr.ng/ml | ALA5238296 | ng.hr.mL-1 | ||||
| 18. | ALA5288241 | B2 | Ratio | > | 48 | ALA5238295 | ||||||
| 19. | ALA5288241 | B2 | Papp | = | 6 | 10^-6 cm/s | ALA5238294 | 10^-6 cm/s | ||||
| 20. | ALA5288241 | B2 | Papp | < | 0 | 10^-6 cm/s | ALA5238293 | 10^-6 cm/s |
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