# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5288342 | 36; ARUK2002821 | INH | = | 63 | % | ALA5260689 | % | Homo sapiens | |||
2. | ALA5288342 | 36; ARUK2002821 | INH | = | 62 | % | ALA5260688 | % | Homo sapiens | |||
3. | ALA5288342 | 36; ARUK2002821 | INH | = | 81.7 | % | ALA5260687 | % | Homo sapiens | |||
4. | ALA5288342 | 36; ARUK2002821 | INH | = | 15.6 | % | ALA5260686 | % | Homo sapiens | |||
5. | ALA5288342 | 36; ARUK2002821 | t1/2 | = | 11 | min | ALA5260685 | hr | ||||
6. | ALA5288342 | 36; ARUK2002821 | Ratio | = | 0.8 | ALA5260684 | ||||||
7. | ALA5288342 | 36; ARUK2002821 | solubility | = | 3 | uM | ALA5260683 | nM | ||||
8. | ALA5288342 | 36; ARUK2002821 | Papp | = | 0.2 | 10^-6 cm/s | ALA5260682 | 10^-6 cm/s | ||||
9. | ALA5288342 | 36; ARUK2002821 | pIC50 | = | 6.6 | ALA5260681 | 6.60 | nM | Homo sapiens | |||
10. | ALA5288342 | 36; ARUK2002821 | pIC50 | < | 4.3 | ALA5260679 | nM | Homo sapiens | ||||
11. | ALA5288342 | 36; ARUK2002821 | pIC50 | = | 8 | ALA5260678 | 8.00 | nM | Homo sapiens | |||
12. | ALA5288342 | 36; ARUK2002821 | INH | = | 4 | % | ALA5260670 | % | Homo sapiens |