# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5288744 | 9 | T/C | = | 0.04 | ALA5252836 | Mus musculus | |||||
2. | ALA5288744 | 9 | T/C | = | 0.22 | ALA5252835 | Mus musculus | |||||
3. | ALA5288744 | 9 | Activity | 0 | ALA5252834 | Non-Toxic | ||||||
4. | ALA5288744 | 9 | Activity | 0 | ALA5252833 | Non-Toxic | ||||||
5. | ALA5288744 | 9 | Activity | 0 | ALA5252832 | Non-Toxic | ||||||
6. | ALA5288744 | 9 | Activity | 0 | ALA5252831 | Non-Toxic | ||||||
7. | ALA5288744 | 9 | Activity | 0 | ALA5252830 | Non-Toxic | ||||||
8. | ALA5288744 | 9 | Activity | 0 | ALA5252829 | Non-Toxic | ||||||
9. | ALA5288744 | 9 | TGI | = | 54 | % | ALA5252828 | % | Mus musculus | |||
10. | ALA5288744 | 9 | TGI | = | 71 | % | ALA5252827 | % | Mus musculus | |||
11. | ALA5288744 | 9 | Activity | 0 | ALA5252825 | Non-Toxic | ||||||
12. | ALA5288744 | 9 | F | = | 5 | % | ALA5252807 | % | ||||
13. | ALA5288744 | 9 | t1/2 | = | 10.1 | hr | ALA5252806 | hr | ||||
14. | ALA5288744 | 9 | AUC/dose | = | 0.67 | umol/l.hr | ALA5252805 | umol/l.hr | ||||
15. | ALA5288744 | 9 | Cmax/dose | = | 0.05 | umol/L | ALA5252804 | umol/L | ||||
16. | ALA5288744 | 9 | Tmax | = | 4 | hr | ALA5252803 | hr | ||||
17. | ALA5288744 | 9 | IC50 | > | 3 | uM | ALA5252799 | nM | Homo sapiens | |||
18. | ALA5288744 | 9 | IC50 | = | 1.7 | nM | ALA5252798 | 8.77 | nM | Homo sapiens | ||
19. | ALA5288744 | 9 | IC50 | > | 10 | uM | ALA5252797 | nM | Mus musculus | |||
20. | ALA5288744 | 9 | IC50 | > | 10 | uM | ALA5252796 | nM | Mus musculus |