# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5290005 | 58; BAY-297 | Fmax | = | 100 | % | ALA5243054 | % | ||||
2. | ALA5290005 | 58; BAY-297 | CLH | = | 0 | L/hr/kg | ALA5243053 | mL.min-1.kg-1 | ||||
3. | ALA5290005 | 58; BAY-297 | IC50 | = | 21.2 | uM | ALA5243052 | 4.67 | nM | Homo sapiens | ||
4. | ALA5290005 | 58; BAY-297 | IC50 | = | 9.5 | uM | ALA5243051 | 5.02 | nM | Homo sapiens | ||
5. | ALA5290005 | 58; BAY-297 | IC50 | = | 30 | uM | ALA5243050 | 4.52 | nM | Homo sapiens | ||
6. | ALA5290005 | 58; BAY-297 | EC50 | = | 18.1 | uM | ALA5243049 | 4.74 | nM | Homo sapiens | ||
7. | ALA5290005 | 58; BAY-297 | INH | 0 | ALA5243048 | Not Active | % | Homo sapiens | ||||
8. | ALA5290005 | 58; BAY-297 | INH | 0 | ALA5243047 | Not Active | % | Homo sapiens | ||||
9. | ALA5290005 | 58; BAY-297 | INH | 0 | ALA5243046 | Not Active | % | Homo sapiens | ||||
10. | ALA5290005 | 58; BAY-297 | INH | 0 | ALA5243045 | Not Active | % | Homo sapiens | ||||
11. | ALA5290005 | 58; BAY-297 | EC50 | = | 1.6 | uM | ALA5243044 | 5.80 | nM | Homo sapiens | ||
12. | ALA5290005 | 58; BAY-297 | EC50 | = | 2.1 | uM | ALA5243043 | 5.68 | nM | Homo sapiens | ||
13. | ALA5290005 | 58; BAY-297 | IC50 | = | 8.35 | uM | ALA5243042 | 5.08 | nM | Homo sapiens | ||
14. | ALA5290005 | 58; BAY-297 | IC50 | = | 10 | uM | ALA5243041 | 5.00 | nM | Homo sapiens | ||
15. | ALA5290005 | 58; BAY-297 | IC50 | > | 10 | uM | ALA5243040 | nM | Homo sapiens | |||
16. | ALA5290005 | 58; BAY-297 | IC50 | = | 3.4 | uM | ALA5243039 | 5.47 | nM | Homo sapiens | ||
17. | ALA5290005 | 58; BAY-297 | IC50 | = | 2.3 | uM | ALA5243038 | 5.64 | nM | Homo sapiens | ||
18. | ALA5290005 | 58; BAY-297 | IC50 | > | 10 | uM | ALA5243037 | nM | Homo sapiens | |||
19. | ALA5290005 | 58; BAY-297 | Drug recovery | = | 18 | % | ALA5243036 | % | ||||
20. | ALA5290005 | 58; BAY-297 | Papp | = | 3.1 | nm/s | ALA5243035 | nm/s |