# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA22969 | vinblastine | Activity | = | 33 | % | ALA5246971 | % | Homo sapiens | |||
2. | ALA22969 | vinblastine | GI50 | = | 37.8 | nM | ALA5236972 | nM | Homo sapiens | |||
3. | ALA22969 | vinblastine | IC50 | = | 0.002 | uM | ALA5231976 | 8.70 | nM | Homo sapiens | ||
4. | ALA22969 | vinblastine | IC50 | = | 0.3 | uM | ALA5130810 | 6.52 | nM | Homo sapiens | ||
5. | ALA22969 | vinblastine | IC50 | = | 0.004 | uM | ALA5130809 | 8.40 | nM | Homo sapiens | ||
6. | ALA22969 | vinblastine | IC50 | = | 1.63 | uM | ALA5130808 | 5.79 | nM | Homo sapiens | ||
7. | ALA22969 | vinblastine | IC50 | = | 0.035 | uM | ALA5130807 | 7.46 | nM | Homo sapiens | ||
8. | ALA22969 | vinblastine | INH | = | 66 | % | ALA5128210 | % | Homo sapiens | |||
9. | ALA22969 | vinblastine | IC50 | = | 0.74 | umol/L | ALA5115598 | 6.13 | nM | Homo sapiens | ||
10. | ALA22969 | vinblastine | IC50 | = | 4.48 | nmol/L | ALA5115596 | 8.35 | nM | Homo sapiens | ||
11. | ALA22969 | vinblastine | IC50 | = | 1.03 | nmol/L | ALA5115595 | 8.99 | nM | Homo sapiens | ||
12. | ALA22969 | vinblastine | IC50 | = | 0.83 | nmol/L | ALA5115594 | 9.08 | nM | |||
13. | ALA22969 | vinblastine | Ratio IC50 | = | 106.8 | ALA4425682 | ||||||
14. | ALA22969 | vinblastine | IC50 | = | 5846 | nM | ALA4425681 | 5.23 | nM | Homo sapiens | ||
15. | ALA22969 | vinblastine | Ratio IC50 | = | 352.4 | ALA4425680 | ||||||
16. | ALA22969 | vinblastine | IC50 | = | 5205 | nM | ALA4425679 | 5.28 | nM | Homo sapiens | ||
17. | ALA22969 | vinblastine | Ratio IC50 | = | 307.3 | ALA4425678 | ||||||
18. | ALA22969 | vinblastine | IC50 | = | 6899 | nM | ALA4425677 | 5.16 | nM | Homo sapiens | ||
19. | ALA22969 | vinblastine | IC50 | = | 22.5 | nM | ALA4425668 | 7.65 | nM | Homo sapiens | ||
20. | ALA22969 | vinblastine | IC50 | = | 54.7 | nM | ALA4425665 | 7.26 | nM | Homo sapiens |