| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA183937 | 4 | EC50 | = | 5.2 | nM | ALA5129913 | 8.28 | nM | Homo sapiens | ||
| 2. | ALA183937 | 4 | EC50 | = | 240 | nM | ALA5129912 | 6.62 | nM | Homo sapiens | ||
| 3. | ALA183937 | 4 | Vdss | = | 11390 | ml/kg | ALA1247341 | L.kg-1 | Rattus norvegicus | |||
| 4. | ALA183937 | 4 | CL | = | 7506 | ml/hr.kg | ALA1247339 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 5. | ALA183937 | 4 | t1/2 | = | 1.3 | hr | ALA1247336 | hr | Rattus norvegicus | |||
| 6. | ALA183937 | 4 | AUC | = | 153 | ng.hr/ml | ALA1247190 | ng.hr.mL-1 | Rattus norvegicus | |||
| 7. | ALA183937 | 4 | IC50 | > | 10000 | nM | ALA1247186 | nM | Rattus norvegicus | |||
| 8. | ALA183937 | 4 | IC50 | = | 240 | nM | ALA1247185 | 6.62 | nM | Homo sapiens | ||
| 9. | ALA183937 | 4 | IC50 | = | 5.2 | nM | ALA1247184 | 8.28 | nM | Homo sapiens | ||
| 10. | ALA183937 | 4 | Selectivity ratio | = | 4 | ALA980893 | ||||||
| 11. | ALA183937 | 4 | EC50 | = | 50 | nM | ALA977369 | 7.30 | nM | Homo sapiens | ||
| 12. | ALA183937 | 4 | Ratio | = | 30 | ALA961710 | ||||||
| 13. | ALA183937 | 4 | IC50 | = | 50 | nM | ALA961709 | 7.30 | nM | Homo sapiens | ||
| 14. | ALA183937 | 4 | EC50 | = | 6.6 | nM | ALA961709 | 8.18 | nM | Homo sapiens | ||
| 15. | ALA183937 | 4 | Ratio EC50 | = | 30 | ALA947999 | ||||||
| 16. | ALA183937 | 4 | EC50 | = | 211 | nM | ALA947998 | 6.68 | nM | Homo sapiens | ||
| 17. | ALA183937 | 4 | EC50 | = | 6.6 | nM | ALA947997 | 8.18 | nM | Homo sapiens | ||
| 18. | ALA183937 | 4 | CL | = | 53.1 | ml/min.kg | ALA867725 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 19. | ALA183937 | 4 | T1/2 | = | 0.97 | hr | ALA867724 | hr | Rattus norvegicus | |||
| 20. | ALA183937 | 4 | AUC | = | 2087 | nM.hr | ALA867218 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus |
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