# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA359803 | 7 | F | = | 50 | % | ALA838660 | % | ||||
2. | ALA359803 | 7 | F | = | 52 | % | ALA838248 | % | Rattus norvegicus | |||
3. | ALA359803 | 7 | AUC | = | 29.56 | ug hr-1 ml-1 | ALA840372 | ng.hr.mL-1 | ||||
4. | ALA359803 | 7 | T1/2 | = | 3.45 | hr | ALA839157 | hr | ||||
5. | ALA359803 | 7 | Cmax | = | 5.58 | ug ml-1 | ALA852888 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
6. | ALA359803 | 7 | Clearance | = | 34 | ml min-1 kg-1 | ALA827498 | mL.min-1.kg-1 | ||||
7. | ALA359803 | 7 | Clearance | = | 6 | ml min-1 kg-1 | ALA828374 | mL.min-1.kg-1 | ||||
8. | ALA359803 | 7 | Clearance | = | 131 | ml min-1 kg-1 | ALA828375 | mL.min-1.kg-1 | ||||
9. | ALA359803 | 7 | ED30 | = | 0.6 | mg kg-1 | ALA833335 | mg kg-1 | Rattus norvegicus | |||
10. | ALA359803 | 7 | IC50 | = | 8.6 | nM | ALA828409 | 8.07 | nM | Homo sapiens |