# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Nutlin-3a | Nutlin-3 | IC50 | = | 0.09 | uM | ALA2156544 | 7.05 | nM | Homo sapiens | ||
2. | Nutlin-3a | Nutlin-3 | IC50 | = | 0.474 | uM | ALA3136838 | 6.32 | nM | Homo sapiens | ||
3. | Nutlin-3a | Nutlin-3 | IC50 | = | 1.9 | uM | ALA3240508 | 5.72 | nM | Homo sapiens | ||
4. | Nutlin-3a | Nutlin-3 | IC50 | = | 0.07 | uM | ALA3240507 | 7.16 | nM | Homo sapiens | ||
5. | Nutlin-3a | Nutlin-3 | permeability | = | 126 | nm/s | ALA3240504 | nm/s | Homo sapiens | |||
6. | Nutlin-3a | Nutlin-3 | Ratio IC50 | = | 30 | ALA3292886 | Homo sapiens | |||||
7. | Nutlin-3a | Nutlin-3 | Activity | 0 | ALA3292885 | Not Active | Homo sapiens | |||||
8. | Nutlin-3a | Nutlin-3 | Ki | = | 0.09 | uM | ALA3294652 | 7.05 | nM | Homo sapiens | ||
9. | Nutlin-3a | Nutlin-3 | IC50 | > | 60 | uM | ALA3222409 | nM | Homo sapiens | |||
10. | Nutlin-3a | Nutlin-3 | IC50 | = | 4.6 | uM | ALA3222408 | 5.34 | nM | Homo sapiens | ||
11. | Nutlin-3a | Nutlin-3 | Kd | < | 1 | uM | ALA3222407 | nM | Homo sapiens | |||
12. | Nutlin-3a | Nutlin-3 | IC50 | = | 90 | nM | ALA3413423 | 7.05 | nM | Homo sapiens | ||
13. | Nutlin-3a | Nutlin-3 | IC50 | = | 1 | uM | ALA3413424 | 6.00 | nM | Homo sapiens | ||
14. | Nutlin-3a | Nutlin-3 | IC50 | = | 1 | uM | ALA3413425 | 6.00 | nM | |||
15. | Nutlin-3a | Nutlin-3 | IC50 | = | 1 | uM | ALA3413426 | 6.00 | nM | Homo sapiens | ||
16. | Nutlin-3a | Nutlin-3 | TGI | = | 90 | % | ALA3413427 | % | Homo sapiens | |||
17. | Nutlin-3a | Nutlin-3 | IC50 | > | 50 | uM | ALA3406262 | nM | Chlorocebus sabaeus | |||
18. | Nutlin-3a | Nutlin-3 | IC50 | > | 50 | uM | ALA3406261 | nM | Homo sapiens | |||
19. | Nutlin-3a | Nutlin-3 | IC50 | = | 11.6 | uM | ALA3406260 | 4.94 | nM | Homo sapiens | ||
20. | Nutlin-3a | Nutlin-3 | IC50 | = | 23.5 | uM | ALA3406259 | 4.63 | nM | Homo sapiens |