# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA195390 | S-(+)-2a | IC50 | = | 172.65 | uM | ALA3271084 | nM | Rattus norvegicus | |||
2. | ALA195390 | S-(+)-2a | Activity | 0 | ALA3271087 | Not Active | Rattus norvegicus | |||||
3. | ALA195390 | S-(+)-2a | Ki | = | 8.21 | uM | ALA3271085 | 5.09 | nM | Rattus norvegicus | ||
4. | ALA195390 | S-(+)-2a | INH | 0 | ALA3271084 | Dose-dependent effect | % | Rattus norvegicus | ||||
5. | ALA195390 | S-(+)-2a | ED50 | = | 0.48 | mg kg-1 | ALA4009970 | mg.kg-1 | Rattus norvegicus | |||
6. | ALA195390 | S-(+)-2a | EC50 | = | 136 | nM | ALA4009968 | 6.87 | nM | |||
7. | ALA195390 | S-(+)-2a | EC50 | = | 142 | nM | ALA4009967 | 6.85 | nM | Rattus norvegicus | ||
8. | ALA195390 | S-(+)-2a | EC50 | = | 74 | nM | ALA4009966 | 7.13 | nM | Rattus norvegicus | ||
9. | ALA195390 | S-(+)-2a | Ki | = | 15800 | nM | ALA4009965 | 4.80 | nM | Rattus norvegicus | ||
10. | ALA195390 | S-(+)-2a | EC50 | = | 0.37 | uM | ALA1930659 | 6.43 | nM | Homo sapiens | ||
11. | ALA195390 | S-(+)-2a | EC50 | = | 16.1 | uM | ALA1930650 | 4.79 | nM | Macaca mulatta | ||
12. | ALA195390 | S-(+)-2a | EC50 | = | 73.7 | uM | ALA1930561 | 4.13 | nM | Homo sapiens | ||
13. | ALA195390 | S-(+)-2a | Vmax | = | 8.4 | ALA873575 | Homo sapiens | |||||
14. | ALA195390 | S-(+)-2a | Km | = | 6.9 | uM | ALA873567 | nM | Homo sapiens | |||
15. | ALA195390 | S-(+)-2a | Vmax | = | 3.8 | 1/min | ALA873573 | 1/min | Homo sapiens | |||
16. | ALA195390 | S-(+)-2a | Km | = | 10.3 | uM | ALA872251 | nM | Homo sapiens | |||
17. | ALA195390 | S-(+)-2a | Vmax | = | 2.4 | ALA873576 | Homo sapiens | |||||
18. | ALA195390 | S-(+)-2a | Km | = | 4.9 | uM | ALA872252 | nM | Homo sapiens | |||
19. | ALA195390 | S-(+)-2a | Vmax | = | 1.2 | 1/min | ALA883679 | 1/min | Homo sapiens | |||
20. | ALA195390 | S-(+)-2a | Km | = | 3.3 | uM | ALA883673 | nM | Homo sapiens |