| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA194564 | 7 | % change | = | -6.9 | % | ALA857460 | % | Rattus norvegicus | |||
| 2. | ALA194564 | 7 | % change | = | -31 | % | ALA857462 | % | Rattus norvegicus | |||
| 3. | ALA194564 | 7 | % change | = | -16 | % | ALA873676 | % | Rattus norvegicus | |||
| 4. | ALA194564 | 7 | C12h | = | 175 | ng g-1 | ALA884603 | ng g-1 | ||||
| 5. | ALA194564 | 7 | Cmax | = | 454 | ng g-1 | ALA880455 | ng g-1 | ||||
| 6. | ALA194564 | 7 | AUC | = | 4.17 | ug .h/g | ALA884578 | ug .h/g | ||||
| 7. | ALA194564 | 7 | AUC | = | 6.35 | ug .h/mL | ALA872382 | ng.hr.mL-1 | ||||
| 8. | ALA194564 | 7 | Inhibition | = | 60 | % | ALA881870 | % | Homo sapiens | |||
| 9. | ALA194564 | 7 | Inhibition | = | 69 | % | ALA881869 | % | Homo sapiens | |||
| 10. | ALA194564 | 7 | Inhibition | = | 75 | % | ALA881869 | % | Homo sapiens | |||
| 11. | ALA194564 | 7 | IC50 | = | 2.25 | uM | ALA882589 | 5.65 | nM | Homo sapiens | ||
| 12. | ALA194564 | 7 | Activity | = | 48 | % | ALA881920 | % | ||||
| 13. | ALA194564 | 7 | T1/2 | = | 4.4 | hr | ALA880473 | hr | ||||
| 14. | ALA194564 | 7 | Cmax | = | 0.2 | ug ml-1 | ALA884612 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 15. | ALA194564 | 7 | AUC | = | 2.66 | ug hr-1 ml-1 | ALA881991 | ng.hr.mL-1 | ||||
| 16. | ALA194564 | 7 | Clp | = | 0.95 | l hr-1 kg-1 | ALA884580 | mL.min-1.kg-1 | ||||
| 17. | ALA194564 | 7 | IC50 | = | 28 | nM | ALA871872 | 7.55 | nM | Homo sapiens | ||
| 18. | ALA194564 | 7 | Cmax | = | 1.6 | ug ml-1 | ALA884621 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 19. | ALA194564 | 7 | T1/2 | = | 3.9 | hr | ALA880478 | hr | ||||
| 20. | ALA194564 | 7 | Activity | = | 19.89 | ug ml-1 | ALA881927 | ug ml-1 |
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