# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA202832 | 7d | IC50 | = | 1.06 | uM | ALA5227658 | 5.97 | nM | |||
2. | ALA202832 | 7d | Kd | = | 0.15 | uM | ALA5227657 | 6.82 | nM | |||
3. | ALA202832 | 7d | Drug uptake | = | 0.74 | nmol/mg | ALA859545 | nmol/mg | Mus musculus | |||
4. | ALA202832 | 7d | Drug uptake | = | 0.54 | nmol/mg | ALA863499 | nmol/mg | Mus musculus | |||
5. | ALA202832 | 7d | Drug uptake | = | 7.8 | nmol/mg | ALA863500 | nmol/mg | Mus musculus | |||
6. | ALA202832 | 7d | Drug uptake | = | 9.4 | nmol/mg | ALA863496 | nmol/mg | Mus musculus | |||
7. | ALA202832 | 7d | Drug uptake | = | 0.66 | nmol/mg | ALA864650 | nmol/mg | Mus musculus | |||
8. | ALA202832 | 7d | Drug uptake | = | 17 | nmol/mg | ALA864647 | nmol/mg | Mus musculus | |||
9. | ALA202832 | 7d | Drug uptake | = | 0.07 | nmol/mg | ALA862824 | nmol/mg | Mus musculus | |||
10. | ALA202832 | 7d | Drug uptake | = | 1.1 | nmol/mg | ALA862821 | nmol/mg | Mus musculus | |||
11. | ALA202832 | 7d | IC50 | = | 3.1 | uM | ALA864027 | 5.51 | nM | Mus musculus | ||
12. | ALA202832 | 7d | IC50 | = | 11 | uM | ALA859860 | 4.96 | nM | Cricetulus griseus | ||
13. | ALA202832 | 7d | Selectivity ratio | = | 0.9 | ALA864028 | ||||||
14. | ALA202832 | 7d | Drug uptake | = | 0.81 | nmol/mg | ALA864640 | nmol/mg | Cricetulus griseus | |||
15. | ALA202832 | 7d | Drug uptake | = | 0.72 | nmol/mg | ALA864639 | nmol/mg | Cricetulus griseus | |||
16. | ALA202832 | 7d | IC50 | = | 23 | uM | ALA864638 | 4.64 | nM | Cricetulus griseus | ||
17. | ALA202832 | 7d | IC50 | = | 23 | uM | ALA864631 | 4.64 | nM | Bos taurus |