# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA201138 | 12 | Inhibition | = | 59 | % | ALA859809 | % | Rattus norvegicus | |||
2. | ALA201138 | 12 | IC50 | = | 0.005 | uM | ALA859578 | 8.30 | nM | Homo sapiens | ||
3. | ALA201138 | 12 | T1/2 | = | 5.5 | hr | ALA859815 | hr | Rattus norvegicus | |||
4. | ALA201138 | 12 | Cz | = | 2.7 | ug ml-1 | ALA859813 | ug ml-1 | Rattus norvegicus | |||
5. | ALA201138 | 12 | tz | = | 24 | hr | ALA859814 | hr | Rattus norvegicus | |||
6. | ALA201138 | 12 | AUC | = | 336.1 | ug.hr/mL | ALA859818 | ng.hr.mL-1 | Rattus norvegicus | |||
7. | ALA201138 | 12 | Papp | = | 6.6 | cm/s | ALA859819 | cm/s | Homo sapiens | |||
8. | ALA201138 | 12 | Tmax | = | 6 | hr | ALA859811 | hr | Rattus norvegicus | |||
9. | ALA201138 | 12 | AUC | = | 314.5 | ug.hr/mL | ALA859817 | ng.hr.mL-1 | Rattus norvegicus | |||
10. | ALA201138 | 12 | Inhibition | 0 | ALA859577 | Not Active | % | Homo sapiens | ||||
11. | ALA201138 | 12 | Inhibition | = | 55 | % | ALA859581 | % | Rattus norvegicus | |||
12. | ALA201138 | 12 | Cmax | = | 22.7 | ug ml-1 | ALA859810 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
13. | ALA201138 | 12 | CL | = | 0.12 | L/hrs.kg | ALA859816 | mL.min-1.kg-1 | Rattus norvegicus |