| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA201914 | rac-34a | AUC | = | 18.5 | uM.hr | ALA886088 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 2. | ALA201914 | rac-34a | t1/2 | = | 3.5 | hr | ALA886087 | hr | Rattus norvegicus | |||
| 3. | ALA201914 | rac-34a | F | = | 39 | % | ALA886086 | % | Rattus norvegicus | |||
| 4. | ALA201914 | rac-34a | Ratio IC50 | = | 76 | ALA886082 | ||||||
| 5. | ALA201914 | rac-34a | IC50 | = | 38 | nM | ALA886081 | 7.42 | nM | Oryctolagus cuniculus | ||
| 6. | ALA201914 | rac-34a | Selectivity ratio | = | 1100 | ALA886080 | ||||||
| 7. | ALA201914 | rac-34a | Selectivity ratio | > | 120000 | ALA886079 | ||||||
| 8. | ALA201914 | rac-34a | Selectivity ratio | = | 880 | ALA886078 | ||||||
| 9. | ALA201914 | rac-34a | IC50 | = | 0.5 | nM | ALA886077 | 9.30 | nM | Oryctolagus cuniculus | ||
| 10. | ALA201914 | rac-34a | IC50 | = | 0.5 | nM | ALA886076 | 9.30 | nM | Homo sapiens | ||
| 11. | ALA201914 | rac-34a | Ratio IC50 | = | 53 | ALA886082 | ||||||
| 12. | ALA201914 | rac-34a | IC50 | = | 16 | nM | ALA886081 | 7.80 | nM | Oryctolagus cuniculus | ||
| 13. | ALA201914 | rac-34a | Selectivity ratio | = | 940 | ALA886080 | ||||||
| 14. | ALA201914 | rac-34a | Selectivity ratio | > | 36000 | ALA886079 | ||||||
| 15. | ALA201914 | rac-34a | Selectivity ratio | = | 780 | ALA886078 | ||||||
| 16. | ALA201914 | rac-34a | IC50 | = | 0.3 | nM | ALA886077 | 9.52 | nM | Oryctolagus cuniculus | ||
| 17. | ALA201914 | rac-34a | IC50 | = | 0.3 | nM | ALA886076 | 9.52 | nM | Homo sapiens | ||
| 18. | ALA201914 | rac-34a | F | = | 53 | % | ALA867017 | % | Rattus norvegicus | |||
| 19. | ALA201914 | rac-34a | IC50 | = | 0.5 | nM | ALA858799 | 9.30 | nM | Oryctolagus cuniculus | ||
| 20. | ALA201914 | rac-34a | CL | = | 15 | ml/min.kg | ALA864080 | mL.min-1.kg-1 | Rattus norvegicus |
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