Activities

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Activities

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#	Name	Compound Key	Action Type	Relation	Activity Value	Units	Assay ID	Assay Description	Assay	Assay Organism
1.	relacatib	10	INH	<=	57	%	ALA1120152		%	Macaca fascicularis
2.	relacatib	10	Activity	=	42	%	ALA1120153		%	Macaca fascicularis
3.	relacatib	10	Activity	=	49	%	ALA1120154		%	Macaca fascicularis
4.	relacatib	10	Selectivity ratio	=	39		ALA1119725
5.	relacatib	10	Selectivity ratio	=	1.65		ALA1119724
6.	relacatib	10	Selectivity ratio	=	317		ALA1119723
7.	relacatib	10	Selectivity ratio	=	39		ALA1120135
8.	relacatib	10	Ki(app)	=	0.041	nM	ALA1119720	10.39	nM	Homo sapiens
9.	relacatib	10	CL	=	19.5	ml/min.kg	ALA1120144		mL.min-1.kg-1	Rattus norvegicus
10.	relacatib	10	Vdss	=	1.79	L/Kg	ALA1120145		L.kg-1	Rattus norvegicus
11.	relacatib	10	F	=	89	%	ALA1120146		%	Rattus norvegicus
12.	relacatib	10	CL	=	11.7	ml/min.kg	ALA1120147		mL.min-1.kg-1	Macaca fascicularis
13.	relacatib	10	Vdss	=	0.95	L/Kg	ALA1120148		L.kg-1	Macaca fascicularis
14.	relacatib	10	F	=	28	%	ALA1120143		%	Macaca fascicularis
15.	relacatib	10	INH	<=	57	%	ALA1120149		%	Macaca fascicularis
16.	relacatib	10	INH	<=	57	%	ALA1120150		%	Macaca fascicularis
17.	relacatib	10	INH	<=	57	%	ALA1120151		%	Macaca fascicularis
18.	relacatib	10	IC50	=	0.5	nM	ALA945079	9.30	nM	Homo sapiens
19.	relacatib	10	IC50	=	8	nM	ALA945093	8.10	nM	Homo sapiens
20.	relacatib	10	IC50	=	2	nM	ALA945092	8.70	nM	Homo sapiens