# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA378379 | 14 | Ratio | = | 0.4 | ALA861182 | Homo sapiens | |||||
2. | ALA378379 | 14 | permeability | = | 11 | %/hr | ALA861181 | %/hr | Homo sapiens | |||
3. | ALA378379 | 14 | permeability | = | 26 | %/hr | ALA861180 | %/hr | Homo sapiens | |||
4. | ALA378379 | 14 | Selectivity ratio | = | 150 | ALA860403 | Homo sapiens | |||||
5. | ALA378379 | 14 | Selectivity ratio | = | 150 | ALA862357 | Homo sapiens | |||||
6. | ALA378379 | 14 | Log D | = | 2.8 | ALA861178 | ||||||
7. | ALA378379 | 14 | pKa | = | 8.8 | ALA861179 | ||||||
8. | ALA378379 | 14 | IC50 | = | 440 | nM | ALA862356 | 6.36 | nM | Homo sapiens | ||
9. | ALA378379 | 14 | IC50 | = | 450 | nM | ALA862305 | 6.35 | nM | Homo sapiens | ||
10. | ALA378379 | 14 | IC50 | = | 3 | nM | ALA862304 | 8.52 | nM | Homo sapiens |