| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA203535 | 18 | INH | = | 90 | % | ALA5144922 | % | ||||
| 2. | ALA203535 | 18 | INH | = | 13 | % | ALA5144921 | % | ||||
| 3. | ALA203535 | 18 | IC50 | = | 23 | uM | ALA5144920 | 4.64 | nM | Homo sapiens | ||
| 4. | ALA203535 | 18 | IC50 | = | 0.67 | uM | ALA5144919 | 6.17 | nM | Homo sapiens | ||
| 5. | ALA203535 | 18 | IC50 | = | 1 | uM | ALA5144918 | 6.00 | nM | Homo sapiens | ||
| 6. | ALA203535 | 18 | IC50 | = | 1 | uM | ALA5144917 | 6.00 | nM | Homo sapiens | ||
| 7. | ALA203535 | 18 | IC50 | = | 180 | nM | ALA1103397 | 6.75 | nM | Homo sapiens | ||
| 8. | ALA203535 | 18 | IC50 | = | 384 | nM | ALA1116944 | 6.42 | nM | Homo sapiens | ||
| 9. | ALA203535 | 18 | IC50 | = | 7 | nM | ALA1116946 | 8.15 | nM | Homo sapiens | ||
| 10. | ALA203535 | 18 | F | = | 16 | % | ALA1103395 | % | Rattus norvegicus | |||
| 11. | ALA203535 | 18 | pIC50 | = | 6.7 | ALA1108472 | 6.70 | nM | Homo sapiens | |||
| 12. | ALA203535 | 18 | pIC50 | = | 8.2 | ALA1108471 | 8.20 | nM | Homo sapiens | |||
| 13. | ALA203535 | 18 | pIC50 | = | 6.4 | ALA1108470 | 6.40 | nM | Homo sapiens | |||
| 14. | ALA203535 | 18 | T1/2 | = | 4.7 | hr | ALA862187 | hr | Rattus norvegicus | |||
| 15. | ALA203535 | 18 | CL | = | 30 | ml/min.kg | ALA862186 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 16. | ALA203535 | 18 | F | = | 16 | % | ALA862185 | % | Rattus norvegicus | |||
| 17. | ALA203535 | 18 | CL | = | 12 | uL/min.mg | ALA862181 | mL.min-1.g-1 | Rattus norvegicus | |||
| 18. | ALA203535 | 18 | permeability | = | 29.9 | ucm/s | ALA862183 | ucm/s | Homo sapiens | |||
| 19. | ALA203535 | 18 | IC50 | = | 180 | nM | ALA862178 | 6.75 | nM | Homo sapiens | ||
| 20. | ALA203535 | 18 | IC50 | = | 384 | nM | ALA862177 | 6.42 | nM | Homo sapiens |
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