| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA427202 | 13 | IC50 | = | 807 | nM | ALA3536559 | 6.09 | nM | Homo sapiens | ||
| 2. | ALA427202 | 13 | IC50 | = | 1011 | nM | ALA3536558 | 6.00 | nM | Homo sapiens | ||
| 3. | ALA427202 | 13 | IC50 | = | 687 | nM | ALA3536557 | 6.16 | nM | Homo sapiens | ||
| 4. | ALA427202 | 13 | IC50 | = | 22 | nM | ALA3536556 | 7.66 | nM | Homo sapiens | ||
| 5. | ALA427202 | 13 | IC50 | = | 20 | nM | ALA3536555 | 7.70 | nM | Homo sapiens | ||
| 6. | ALA427202 | 13 | Km | = | 0.7 | uM | ALA3536554 | nM | Homo sapiens | |||
| 7. | ALA427202 | 13 | Km | = | 0.7 | uM | ALA3541059 | nM | ||||
| 8. | ALA427202 | 13 | Km | = | 0.7 | uM | ALA3541058 | nM | Rattus norvegicus | |||
| 9. | ALA427202 | 13 | AUCt | = | 0.4 | ug.hr/ml | ALA3541057 | ng.hr.mL-1 | Homo sapiens | |||
| 10. | ALA427202 | 13 | Tmax | = | 5 | hr | ALA3532265 | hr | Homo sapiens | |||
| 11. | ALA427202 | 13 | Cmax | = | 0.05 | ug ml-1 | ALA3532264 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Homo sapiens | ||
| 12. | ALA427202 | 13 | AUCt | = | 2.7 | ug.hr/ml | ALA3532260 | ng.hr.mL-1 | Macaca fascicularis | |||
| 13. | ALA427202 | 13 | Tmax | = | 4 | hr | ALA3532259 | hr | Macaca fascicularis | |||
| 14. | ALA427202 | 13 | Cmax | = | 0.5 | ug ml-1 | ALA3532258 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Macaca fascicularis | ||
| 15. | ALA427202 | 13 | AUCt | = | 7.2 | ug.hr/ml | ALA3532254 | ng.hr.mL-1 | Rattus norvegicus | |||
| 16. | ALA427202 | 13 | Tmax | = | 2 | hr | ALA3532253 | hr | Rattus norvegicus | |||
| 17. | ALA427202 | 13 | Cmax | = | 2.6 | ug ml-1 | ALA3532252 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 18. | ALA427202 | 13 | Drug metabolism | 0 | ALA3531904 | metabolite_not_detected | Homo sapiens | |||||
| 19. | ALA427202 | 13 | Drug metabolism | 0 | ALA3531903 | metabolite_not_detected | ||||||
| 20. | ALA427202 | 13 | Drug metabolism | 0 | ALA3534831 | metabolite_not_detected | Rattus norvegicus |
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