# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA24461 | 4, BMS-193884 | Ki | = | 1.9 | uM | ALA4426332 | 5.72 | nM | Rattus norvegicus | ||
2. | ALA24461 | 4, BMS-193884 | Ki | = | 1.4 | nM | ALA4426326 | 8.85 | nM | Rattus norvegicus | ||
3. | ALA24461 | 4, BMS-193884 | Ki | > | 10000 | nM | ALA2184411 | nM | Homo sapiens | |||
4. | ALA24461 | 4, BMS-193884 | Ki | = | 1.4 | nM | ALA2184410 | 8.85 | nM | Homo sapiens | ||
5. | ALA24461 | 4, BMS-193884 | Activity | = | 250 | nm/s | ALA838161 | nm/s | Homo sapiens | |||
6. | ALA24461 | 4, BMS-193884 | Activity | = | 9700 | AUC units | ALA826887 | AUC units | Rattus norvegicus | |||
7. | ALA24461 | 4, BMS-193884 | Activity | 0 | AUC units | ALA835823 | Not Active | Rattus norvegicus | ||||
8. | ALA24461 | 4, BMS-193884 | Ki | = | 18700 | nM | ALA673226 | 4.73 | nM | Homo sapiens | ||
9. | ALA24461 | 4, BMS-193884 | KB | = | 19 | nM | ALA768052 | nM | Oryctolagus cuniculus | |||
10. | ALA24461 | 4, BMS-193884 | Ki | = | 1.4 | nM | ALA681520 | 8.85 | nM | Homo sapiens | ||
11. | ALA24461 | 4, BMS-193884 | F | = | 71 | % | ALA633870 | % | ||||
12. | ALA24461 | 4, BMS-193884 | T1/2 | = | 8.7 | hr | ALA877627 | hr | ||||
13. | ALA24461 | 4, BMS-193884 | Cmax | = | 180 | uM | ALA637989 | nM | ||||
14. | ALA24461 | 4, BMS-193884 | T max | = | 2.4 | hr | ALA642686 | hr | ||||
15. | ALA24461 | 4, BMS-193884 | AUC | = | 704 | uM kg-1 | ALA638335 | uM kg-1 | ||||
16. | ALA24461 | 4, BMS-193884 | MRT | = | 2.7 | hr | ALA638559 | hr | ||||
17. | ALA24461 | 4, BMS-193884 | T1/2 | = | 8.3 | hr | ALA633886 | hr | ||||
18. | ALA24461 | 4, BMS-193884 | Vss | = | 0.13 | l kg-1 | ALA642530 | L.kg-1 | ||||
19. | ALA24461 | 4, BMS-193884 | Cl | = | 0.86 | ml min-1 kg-1 | ALA644244 | mL.min-1.kg-1 | ||||
20. | ALA24461 | 4, BMS-193884 | AUC | = | 1000 | uM kg-1 | ALA638333 | uM kg-1 |