# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA378376 | 16c | Ki | = | 2 | nM | ALA5242762 | 8.70 | nM | Homo sapiens | ||
2. | ALA378376 | 16c | IC50 | = | 2 | nM | ALA5242761 | 8.70 | nM | Homo sapiens | ||
3. | ALA378376 | 16c | EC50 | = | 0.5 | nM | ALA1119848 | 9.30 | nM | Rattus norvegicus | ||
4. | ALA378376 | 16c | Activity | = | 102 | % | ALA1117753 | % | Rattus norvegicus | |||
5. | ALA378376 | 16c | CL | = | 70 | ml/min.kg | ALA1120164 | mL.min-1.kg-1 | Rattus norvegicus | |||
6. | ALA378376 | 16c | F | = | 1 | % | ALA1120166 | % | Rattus norvegicus | |||
7. | ALA378376 | 16c | t1/2 | = | 0.2 | hr | ALA1120165 | hr | Rattus norvegicus | |||
8. | ALA378376 | 16c | Activity | = | 22.9 | % | ALA1117755 | % | Rattus norvegicus | |||
9. | ALA378376 | 16c | IC50 | = | 483 | nM | ALA1120704 | 6.32 | nM | Rattus norvegicus | ||
10. | ALA378376 | 16c | IC50 | = | 6 | nM | ALA1120705 | 8.22 | nM | Rattus norvegicus | ||
11. | ALA378376 | 16c | Activity | = | 43.27 | % | ALA859918 | % | Rattus norvegicus | |||
12. | ALA378376 | 16c | Activity | = | 35.76 | % | ALA859917 | % | Rattus norvegicus | |||
13. | ALA378376 | 16c | Activity | = | 62.57 | % | ALA859914 | % | Rattus norvegicus | |||
14. | ALA378376 | 16c | Activity | = | 52.69 | % | ALA859913 | % | Rattus norvegicus | |||
15. | ALA378376 | 16c | Activity | = | 41.77 | % | ALA859910 | % | Rattus norvegicus | |||
16. | ALA378376 | 16c | Activity | = | 34.31 | % | ALA859909 | % | Rattus norvegicus | |||
17. | ALA378376 | 16c | Activity | = | 26.36 | % | ALA859864 | % | Rattus norvegicus | |||
18. | ALA378376 | 16c | Activity | = | 22.88 | % | ALA861031 | % | Rattus norvegicus | |||
19. | ALA378376 | 16c | Activity | = | 23.72 | % | ALA861028 | % | Rattus norvegicus | |||
20. | ALA378376 | 16c | Activity | = | 20.59 | % | ALA861027 | % | Rattus norvegicus |