| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA27979 | A6, A-349821 | pKi | = | 8.8 | ALA2154939 | 8.80 | nM | Homo sapiens | |||
| 2. | ALA27979 | A6, A-349821 | pKi | = | 9.4 | ALA2154938 | 9.40 | nM | Rattus norvegicus | |||
| 3. | ALA27979 | A6, A-349821 | Ki | = | 12 | nM | ALA986460 | 7.92 | nM | Homo sapiens | ||
| 4. | ALA27979 | A6, A-349821 | Ki | = | 2 | nM | ALA1008299 | 8.70 | nM | Homo sapiens | ||
| 5. | ALA27979 | A6, A-349821 | Log Ki | = | -9.31 | ALA889157 | 9.31 | nM | Homo sapiens | |||
| 6. | ALA27979 | A6, A-349821 | Log Ki | = | -8.78 | ALA887978 | 8.78 | nM | Rattus norvegicus | |||
| 7. | ALA27979 | A6, A-349821 | F | = | 33 | % | ALA618876 | % | Canis lupus familiaris | |||
| 8. | ALA27979 | A6, A-349821 | Cmax | = | 0.31 | ug ml-1 | ALA619614 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Canis lupus familiaris | ||
| 9. | ALA27979 | A6, A-349821 | T1/2 | = | 2.6 | hr | ALA624303 | hr | Canis lupus familiaris | |||
| 10. | ALA27979 | A6, A-349821 | Clp | = | 0.6 | l hr-1 kg-1 | ALA624464 | mL.min-1.kg-1 | Canis lupus familiaris | |||
| 11. | ALA27979 | A6, A-349821 | Cmax | = | 0.17 | ug ml-1 | ALA620930 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 12. | ALA27979 | A6, A-349821 | Vbeta | = | 7.5 | l kg-1 | ALA620960 | L.kg-1 | ||||
| 13. | ALA27979 | A6, A-349821 | T1/2 | = | 5.3 | hr | ALA618287 | hr | ||||
| 14. | ALA27979 | A6, A-349821 | Clp | = | 1 | l hr-1 kg-1 | ALA621476 | mL.min-1.kg-1 | ||||
| 15. | ALA27979 | A6, A-349821 | F | = | 78 | % | ALA620934 | % | ||||
| 16. | ALA27979 | A6, A-349821 | pA2 | = | 9.47 | ALA857043 | 9.47 | nM | Cavia porcellus | |||
| 17. | ALA27979 | A6, A-349821 | pKb | = | 9.23 | ALA697532 | Rattus norvegicus | |||||
| 18. | ALA27979 | A6, A-349821 | pA2 | = | 8.71 | ALA697529 | 8.71 | nM | Rattus norvegicus | |||
| 19. | ALA27979 | A6, A-349821 | pA2 | = | 8.67 | ALA694887 | 8.67 | nM | Homo sapiens | |||
| 20. | ALA27979 | A6, A-349821 | Log Ki | = | -5 | ALA858410 | 5.00 | nM | Homo sapiens |
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