# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA204997 | 2 | AUC | = | 1.021 | uM.hr | ALA4624403 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
2. | ALA204997 | 2 | IC50 | = | 249 | nM | ALA4624398 | 6.60 | nM | Homo sapiens | ||
3. | ALA204997 | 2 | IC50 | = | 950 | nM | ALA4624397 | 6.02 | nM | Homo sapiens | ||
4. | ALA204997 | 2 | Ratio IC50 | = | 13 | ALA4624396 | ||||||
5. | ALA204997 | 2 | IC50 | = | 700 | nM | ALA4624395 | 6.16 | nM | Homo sapiens | ||
6. | ALA204997 | 2 | IC50 | = | 53 | nM | ALA4624394 | 7.28 | nM | Homo sapiens | ||
7. | ALA204997 | 2 | PPB | 88.11 | % | ALA3301366 | % | |||||
8. | ALA204997 | 2 | Selectivity ratio | = | 44 | ALA858906 | ||||||
9. | ALA204997 | 2 | Selectivity ratio | = | 96 | ALA869025 | Homo sapiens | |||||
10. | ALA204997 | 2 | Selectivity ratio | = | 36 | ALA869024 | ||||||
11. | ALA204997 | 2 | Selectivity ratio | = | 813 | ALA869023 | ||||||
12. | ALA204997 | 2 | 2PT | = | 14.5 | uM | ALA869022 | uM | Homo sapiens | |||
13. | ALA204997 | 2 | 2aPTT | = | 2.64 | uM | ALA869021 | uM | Homo sapiens | |||
14. | ALA204997 | 2 | Ki | = | 0.05 | uM | ALA869020 | 7.30 | nM | Homo sapiens |