# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA8389 | 1b | pA2 | = | 6.81 | ALA3279114 | 6.81 | nM | Rattus norvegicus | |||
2. | ALA8389 | 1b | log(activity) | = | 1.26 | ALA3258805 | Homo sapiens | |||||
3. | ALA8389 | 1b | Ki | = | 57.9 | nM | ALA4009956 | 7.24 | nM | Homo sapiens | ||
4. | ALA8389 | 1b | Ki | = | 81 | nM | ALA4009955 | 7.09 | nM | Rattus norvegicus | ||
5. | ALA8389 | 1b | Ki | = | 1200 | nM | ALA4009954 | 5.92 | nM | Rattus norvegicus | ||
6. | ALA8389 | 1b | Ki | = | 1200 | nM | ALA994216 | 5.92 | nM | Homo sapiens | ||
7. | ALA8389 | 1b | Activity | = | 10 | ALA700102 | Homo sapiens | |||||
8. | ALA8389 | 1b | KDNB | = | 1.7 | ALA843592 | ||||||
9. | ALA8389 | 1b | pA2 | = | 6.81 | ALA858114 | 6.81 | nM | Rattus norvegicus | |||
10. | ALA8389 | 1b | Relative activity | = | 11.8 | ALA773948 | Oryctolagus cuniculus | |||||
11. | ALA8389 | 1b | Relative activity | = | 17 | ALA878435 | Homo sapiens | |||||
12. | ALA8389 | 1b | logP | = | 1.1 | ALA633218 | ||||||
13. | ALA8389 | 1b | logP | = | 1.74 | ALA633218 | ||||||
14. | ALA8389 | 1b | Ki | = | 1200 | nM | ALA621544 | 5.92 | nM | Rattus norvegicus | ||
15. | ALA8389 | 1b | ED50 | = | 3.59 | mg kg-1 | ALA782002 | mg.kg-1 | Rattus norvegicus | |||
16. | ALA8389 | 1b | Log activity | = | 1.301 | ALA631963 | Homo sapiens | |||||
17. | ALA8389 | 1b | Activity | = | 20 | MU | ALA696016 | MU | Homo sapiens | |||
18. | ALA8389 | 1b | Selectivity | = | 0.5 | ALA851510 | Rattus norvegicus | |||||
19. | ALA8389 | 1b | Ki | = | 1250 | nM | ALA617438 | 5.90 | nM | Rattus norvegicus | ||
20. | ALA8389 | 1b | Ki | = | 2666 | nM | ALA616834 | 5.57 | nM | Rattus norvegicus |