# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA212041 | 1h | EC50 | = | 0.13 | uM | ALA866639 | 6.89 | nM | Mus musculus | ||
2. | ALA212041 | 1h | EC50 | = | 0.24 | uM | ALA866796 | 6.62 | nM | Mus musculus | ||
3. | ALA212041 | 1h | Efficacy | = | 76 | % | ALA866797 | % | Mus musculus | |||
4. | ALA212041 | 1h | EC50 | = | 103 | uM | ALA866793 | nM | Rattus norvegicus | |||
5. | ALA212041 | 1h | EC50 | = | 0.18 | uM | ALA866794 | 6.75 | nM | Homo sapiens | ||
6. | ALA212041 | 1h | EC50 | = | 0.04 | uM | ALA866792 | 7.40 | nM | Rattus norvegicus | ||
7. | ALA212041 | 1h | Inhibition | = | 86 | % | ALA864946 | % | Rattus norvegicus | |||
8. | ALA212041 | 1h | ID50 | = | 4 | mg kg-1 | ALA864947 | mg.kg-1 | Rattus norvegicus | |||
9. | ALA212041 | 1h | IC50 | = | 360 | uM | ALA864945 | nM | Homo sapiens | |||
10. | ALA212041 | 1h | IC50 | = | 0.081 | uM | ALA864943 | 7.09 | nM | Homo sapiens | ||
11. | ALA212041 | 1h | Cmax | = | 2587 | ng/ml | ALA869726 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
12. | ALA212041 | 1h | Tmax | = | 15 | min | ALA869727 | hr | Rattus norvegicus | |||
13. | ALA212041 | 1h | F | = | 82 | % | ALA869728 | % | Rattus norvegicus | |||
14. | ALA212041 | 1h | CL | = | 7.3 | ml/min.kg | ALA869729 | mL.min-1.kg-1 | Rattus norvegicus | |||
15. | ALA212041 | 1h | T1/2 | = | 52 | min | ALA869730 | hr | Rattus norvegicus |