# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA212479 | 1c | EC50 | = | 0.4 | uM | ALA866639 | 6.40 | nM | Mus musculus | ||
2. | ALA212479 | 1c | EC50 | = | 1.4 | uM | ALA866796 | 5.85 | nM | Mus musculus | ||
3. | ALA212479 | 1c | Efficacy | = | 76 | % | ALA866797 | % | Mus musculus | |||
4. | ALA212479 | 1c | EC50 | = | 40 | uM | ALA866793 | 4.40 | nM | Rattus norvegicus | ||
5. | ALA212479 | 1c | EC50 | = | 0.53 | uM | ALA866794 | 6.28 | nM | Homo sapiens | ||
6. | ALA212479 | 1c | EC50 | = | 0.16 | uM | ALA866792 | 6.80 | nM | Rattus norvegicus | ||
7. | ALA212479 | 1c | Inhibition | = | 90 | % | ALA864946 | % | Rattus norvegicus | |||
8. | ALA212479 | 1c | ID50 | = | 8 | mg kg-1 | ALA864947 | mg.kg-1 | Rattus norvegicus | |||
9. | ALA212479 | 1c | Cmax | = | 533 | ng/ml | ALA868562 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
10. | ALA212479 | 1c | Tmax | = | 30 | min | ALA868563 | hr | Rattus norvegicus | |||
11. | ALA212479 | 1c | F | = | 70 | % | ALA868564 | % | Rattus norvegicus | |||
12. | ALA212479 | 1c | CL | = | 5 | ml/min.kg | ALA868565 | mL.min-1.kg-1 | Rattus norvegicus | |||
13. | ALA212479 | 1c | T1/2 | = | 330 | min | ALA868566 | hr | Rattus norvegicus |