# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA210749 | 1m | EC50 | = | 0.14 | uM | ALA866639 | 6.85 | nM | Mus musculus | ||
2. | ALA210749 | 1m | EC50 | = | 0.31 | uM | ALA866796 | 6.51 | nM | Mus musculus | ||
3. | ALA210749 | 1m | Efficacy | = | 81 | % | ALA866797 | % | Mus musculus | |||
4. | ALA210749 | 1m | EC50 | = | 133 | uM | ALA866793 | nM | Rattus norvegicus | |||
5. | ALA210749 | 1m | EC50 | = | 0.16 | uM | ALA866794 | 6.80 | nM | Homo sapiens | ||
6. | ALA210749 | 1m | EC50 | = | 0.02 | uM | ALA866792 | 7.70 | nM | Rattus norvegicus | ||
7. | ALA210749 | 1m | Inhibition | = | 97 | % | ALA864946 | % | Rattus norvegicus | |||
8. | ALA210749 | 1m | ID50 | < | 3 | mg kg-1 | ALA864947 | mg.kg-1 | Rattus norvegicus | |||
9. | ALA210749 | 1m | Cp | = | 340 | ng/ml | ALA867922 | ng/ml | Rattus norvegicus | |||
10. | ALA210749 | 1m | Cmax | = | 885 | ng/ml | ALA868567 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
11. | ALA210749 | 1m | Tmax | = | 90 | min | ALA868568 | hr | Rattus norvegicus | |||
12. | ALA210749 | 1m | F | = | 96 | % | ALA868569 | % | Rattus norvegicus | |||
13. | ALA210749 | 1m | CL | = | 15 | ml/min.kg | ALA868570 | mL.min-1.kg-1 | Rattus norvegicus | |||
14. | ALA210749 | 1m | T1/2 | = | 156 | min | ALA868571 | hr | Rattus norvegicus |