| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA378763 | R-13 | F | = | 103 | % | ALA914059 | % | Rattus norvegicus | |||
| 2. | ALA378763 | R-13 | Fu | = | 0.106 | ALA914058 | ||||||
| 3. | ALA378763 | R-13 | t1/2 | = | 1.7 | hr | ALA914057 | hr | Rattus norvegicus | |||
| 4. | ALA378763 | R-13 | Vdss | = | 0.44 | L/Kg | ALA914056 | L.kg-1 | Rattus norvegicus | |||
| 5. | ALA378763 | R-13 | CL | = | 3 | ml/min.kg | ALA914055 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 6. | ALA378763 | R-13 | IC50 | 0 | ALA914054 | Not Determined | ||||||
| 7. | ALA378763 | R-13 | IC50 | = | 31.8 | nM | ALA914053 | 7.50 | nM | Homo sapiens | ||
| 8. | ALA378763 | R-13 | IC50 | = | 19.7 | nM | ALA914052 | 7.71 | nM | Homo sapiens | ||
| 9. | ALA378763 | R-13 | IC50 | = | 10.2 | nM | ALA914051 | 7.99 | nM | Oryctolagus cuniculus | ||
| 10. | ALA378763 | R-13 | IC50 | = | 14.3 | nM | ALA914050 | 7.84 | nM | Rattus norvegicus | ||
| 11. | ALA378763 | R-13 | IC50 | = | 18.9 | nM | ALA914049 | 7.72 | nM | Homo sapiens | ||
| 12. | ALA378763 | R-13 | Papp | = | 14 | ucm/s | ALA914048 | ucm/s | Homo sapiens | |||
| 13. | ALA378763 | R-13 | Papp | = | 9 | ucm/s | ALA914047 | ucm/s | Homo sapiens | |||
| 14. | ALA378763 | R-13 | t1/2 | > | 120 | min | ALA914046 | hr | Homo sapiens | |||
| 15. | ALA378763 | R-13 | PPB | = | 97.9 | % | ALA914045 | % | Rattus norvegicus | |||
| 16. | ALA378763 | R-13 | Log D | = | 0.5 | ALA914044 | ||||||
| 17. | ALA378763 | R-13 | Activity | > | 3 | uM | ALA914043 | uM | Homo sapiens | |||
| 18. | ALA378763 | R-13 | Activity | > | 3 | uM | ALA914042 | uM | ||||
| 19. | ALA378763 | R-13 | IC50 | = | 23.7 | nM | ALA914041 | 7.62 | nM | |||
| 20. | ALA378763 | R-13 | IC50 | > | 3 | uM | ALA862884 | nM | Homo sapiens |
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