| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA385587 | 24 | PT | = | 5 | uM | ALA907292 | uM | Rattus norvegicus | |||
| 2. | ALA385587 | 24 | Ki | = | 6 | nM | ALA907291 | 8.22 | nM | Homo sapiens | ||
| 3. | ALA385587 | 24 | Ki | = | 6 | nM | ALA1273257 | 8.22 | nM | Homo sapiens | ||
| 4. | ALA385587 | 24 | 2aPTT | = | 5.4 | uM | ALA1273285 | uM | ||||
| 5. | ALA385587 | 24 | t1/2 | = | 0.57 | hr | ALA918013 | hr | Rattus norvegicus | |||
| 6. | ALA385587 | 24 | Ratio IC50 | > | 300 | ALA918012 | ||||||
| 7. | ALA385587 | 24 | Ratio Ki | > | 1000 | ALA918606 | ||||||
| 8. | ALA385587 | 24 | Ratio Ki | > | 1000 | ALA918605 | ||||||
| 9. | ALA385587 | 24 | Ratio Ki | > | 1000 | ALA918604 | ||||||
| 10. | ALA385587 | 24 | Ratio Ki | > | 4500 | ALA918603 | ||||||
| 11. | ALA385587 | 24 | Ratio Ki | > | 4500 | ALA918602 | ||||||
| 12. | ALA385587 | 24 | Ratio Ki | = | 37 | ALA918601 | ||||||
| 13. | ALA385587 | 24 | Activity | = | 79 | % | ALA918600 | % | ||||
| 14. | ALA385587 | 24 | Log D | = | 1.79 | ALA918599 | ||||||
| 15. | ALA385587 | 24 | Ki | = | 6 | nM | ALA918598 | 8.22 | nM | Homo sapiens | ||
| 16. | ALA385587 | 24 | Cp | = | 3 | ml/min.kg | ALA918014 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 17. | ALA385587 | 24 | Vss | = | 0.17 | L/Kg | ALA918015 | L.kg-1 | Rattus norvegicus | |||
| 18. | ALA385587 | 24 | F | = | 69 | % | ALA918016 | % | Rattus norvegicus | |||
| 19. | ALA385587 | 24 | Ki | = | 6 | nM | ALA862916 | 8.22 | nM | Homo sapiens | ||
| 20. | ALA385587 | 24 | Log D | = | 2.2 | ALA862917 |
The page will load shortly, Thanks for your patience!