# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA212907 | 12 | Ki | = | 0.8 | nM | ALA853454 | 9.10 | nM | Homo sapiens | ||
2. | ALA212907 | 12 | Ki | = | 190 | nM | ALA866100 | 6.72 | nM | Homo sapiens | ||
3. | ALA212907 | 12 | Ki | = | 18000 | nM | ALA866101 | 4.75 | nM | Homo sapiens | ||
4. | ALA212907 | 12 | Ki | = | 5600 | nM | ALA866102 | 5.25 | nM | Homo sapiens | ||
5. | ALA212907 | 12 | IC50 | = | 349 | nM | ALA866103 | 6.46 | nM | |||
6. | ALA212907 | 12 | Selectivity ratio | = | 237 | ALA866105 | Homo sapiens | |||||
7. | ALA212907 | 12 | Selectivity ratio | = | 22500 | ALA866106 | Homo sapiens | |||||
8. | ALA212907 | 12 | Selectivity ratio | = | 7000 | ALA866107 | Homo sapiens | |||||
9. | ALA212907 | 12 | Vss | = | 4.3 | L/Kg | ALA864901 | L.kg-1 | Rattus norvegicus | |||
10. | ALA212907 | 12 | MRT | = | 176 | min | ALA864893 | hr | Rattus norvegicus | |||
11. | ALA212907 | 12 | AUC | = | 560 | uM.min | ALA864898 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
12. | ALA212907 | 12 | CL | = | 25 | ml/min.kg | ALA864894 | mL.min-1.kg-1 | Rattus norvegicus | |||
13. | ALA212907 | 12 | Tmax | = | 200 | min | ALA864897 | hr | Rattus norvegicus | |||
14. | ALA212907 | 12 | F | = | 85 | % | ALA864900 | % | Rattus norvegicus | |||
15. | ALA212907 | 12 | T1/2 | = | 3.9 | hr | ALA864899 | hr | Rattus norvegicus | |||
16. | ALA212907 | 12 | Cmax | = | 1.1 | mM | ALA864896 | nM | Rattus norvegicus |