| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA212968 | 75 | IC50 | = | 1.8 | nM | ALA868607 | 8.74 | nM | Homo sapiens | ||
| 2. | ALA212968 | 75 | IC50 | = | 63 | nM | ALA868608 | 7.20 | nM | Homo sapiens | ||
| 3. | ALA212968 | 75 | IC50 | = | 8.3 | nM | ALA867926 | 8.08 | nM | Homo sapiens | ||
| 4. | ALA212968 | 75 | CL | = | 3 | ml/min.kg | ALA868606 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 5. | ALA212968 | 75 | Vdss | = | 0.6 | L/Kg | ALA867928 | L.kg-1 | Rattus norvegicus | |||
| 6. | ALA212968 | 75 | T1/2 | = | 2.6 | hr | ALA867929 | hr | Rattus norvegicus | |||
| 7. | ALA212968 | 75 | F | = | 54 | % | ALA867930 | % | Rattus norvegicus | |||
| 8. | ALA212968 | 75 | CL | = | 3.4 | ml/min.kg | ALA867931 | mL.min-1.kg-1 | Macaca mulatta | |||
| 9. | ALA212968 | 75 | Vdss | = | 1.2 | L/Kg | ALA867932 | L.kg-1 | Macaca mulatta | |||
| 10. | ALA212968 | 75 | T1/2 | = | 5.2 | hr | ALA867933 | hr | Macaca mulatta | |||
| 11. | ALA212968 | 75 | F | = | 66 | % | ALA867934 | % | Macaca mulatta | |||
| 12. | ALA212968 | 75 | Inhibition | = | 5.9 | % | ALA867936 | % | Homo sapiens | |||
| 13. | ALA212968 | 75 | ED50 | = | 0.1 | mg kg-1 | ALA867942 | mg.kg-1 | Rattus norvegicus | |||
| 14. | ALA212968 | 75 | IC50 | > | 10 | uM | ALA867948 | nM | Homo sapiens | |||
| 15. | ALA212968 | 75 | IC50 | > | 10 | uM | ALA867945 | nM | Homo sapiens | |||
| 16. | ALA212968 | 75 | IC50 | > | 10 | uM | ALA867949 | nM | Homo sapiens | |||
| 17. | ALA212968 | 75 | IC50 | > | 10 | uM | ALA869200 | nM | Homo sapiens | |||
| 18. | ALA212968 | 75 | IC50 | > | 10 | uM | ALA869136 | nM | Homo sapiens | |||
| 19. | ALA212968 | 75 | IC50 | > | 10 | uM | ALA869137 | nM | Homo sapiens | |||
| 20. | ALA212968 | 75 | IC50 | > | 10 | uM | ALA869138 | nM | Homo sapiens |
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