# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA212912 | 28 | Activity | 0 | ALA870478 | Antagonist | Homo sapiens | |||||
2. | ALA212912 | 28 | Ratio Ki | = | 44 | ALA911525 | Homo sapiens | |||||
3. | ALA212912 | 28 | Ki | = | 181 | nM | ALA911524 | 6.74 | nM | Homo sapiens | ||
4. | ALA212912 | 28 | Ki | = | 4.1 | nM | ALA911523 | 8.39 | nM | Homo sapiens | ||
5. | ALA212912 | 28 | Ki | = | 73 | nM | ALA870479 | 7.14 | nM | Homo sapiens | ||
6. | ALA212912 | 28 | Kb | = | 2.8 | nM | ALA870478 | nM | Homo sapiens | |||
7. | ALA212912 | 28 | Ki | = | 455 | nM | ALA870476 | 6.34 | nM | Homo sapiens | ||
8. | ALA212912 | 28 | Ki | = | 1 | nM | ALA870475 | 9.00 | nM | Homo sapiens | ||
9. | ALA212912 | 28 | Ki | = | 181 | nM | ALA870474 | 6.74 | nM | Homo sapiens | ||
10. | ALA212912 | 28 | Ki | = | 870 | nM | ALA870473 | 6.06 | nM | Homo sapiens | ||
11. | ALA212912 | 28 | Tmax | = | 1 | hr | ALA870472 | hr | Rattus norvegicus | |||
12. | ALA212912 | 28 | Cmax | = | 821 | ng/ml | ALA870471 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
13. | ALA212912 | 28 | AUC | = | 2656 | ng.hr/ml | ALA870470 | ng.hr.mL-1 | Rattus norvegicus | |||
14. | ALA212912 | 28 | Ratio Ki | = | 45 | ALA870469 | Homo sapiens | |||||
15. | ALA212912 | 28 | Ki | = | 181 | nM | ALA870468 | 6.74 | nM | Homo sapiens | ||
16. | ALA212912 | 28 | Ki | = | 4 | nM | ALA870467 | 8.40 | nM | Homo sapiens |