# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA213330 | 12c | T1/2 | = | 9.5 | min | ALA910298 | hr | Rattus norvegicus | |||
2. | ALA213330 | 12c | T1/2 | = | 9.4 | min | ALA910297 | hr | Mus musculus | |||
3. | ALA213330 | 12c | Papp | = | 0.4 | ucm/s | ALA910296 | ucm/s | Homo sapiens | |||
4. | ALA213330 | 12c | Selectivity ratio | > | 125 | ALA910295 | Plasmodium falciparum | |||||
5. | ALA213330 | 12c | IC50 | > | 1000 | nM | ALA910294 | nM | Rattus norvegicus | |||
6. | ALA213330 | 12c | IC50 | = | 8 | nM | ALA910293 | 8.10 | nM | Plasmodium falciparum | ||
7. | ALA213330 | 12c | ED50 | = | 2600 | nM | ALA910292 | 5.58 | nM | Plasmodium falciparum | ||
8. | ALA213330 | 12c | ED50 | = | 2500 | nM | ALA910874 | 5.60 | nM | Plasmodium falciparum | ||
9. | ALA213330 | 12c | Inhibition | = | 49 | % | ALA910873 | % | Plasmodium falciparum | |||
10. | ALA213330 | 12c | Inhibition | = | 85 | % | ALA909787 | % | Plasmodium falciparum |