# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA224754 | 14 | Activity | 0 | ALA1006228 | Active | ||||||
2. | ALA224754 | 14 | Activity | 0 | ALA1006225 | Active | ||||||
3. | ALA224754 | 14 | Activity | = | 46 | nM | ALA1005444 | nM | ||||
4. | ALA224754 | 14 | Activity | = | 176 | nM | ALA1005443 | nM | ||||
5. | ALA224754 | 14 | Activity | 0 | ALA1006222 | Active | ||||||
6. | ALA224754 | 14 | Tm | = | 83 | degrees C | ALA1006220 | degrees C | ||||
7. | ALA224754 | 14 | Tm | = | 64 | degrees C | ALA1006221 | degrees C | ||||
8. | ALA224754 | 14 | Activity | 0 | ALA1005442 | Active | ||||||
9. | ALA224754 | 14 | Activity | 0 | ALA1005441 | Not Active | ||||||
10. | ALA224754 | 14 | Activity | 0 | ALA1005440 | Not Active | ||||||
11. | ALA224754 | 14 | Activity | 0 | ALA1003665 | Not Active | ||||||
12. | ALA224754 | 14 | Activity | 0 | ALA1006230 | Not Active | ||||||
13. | ALA224754 | 14 | Activity | 0 | ALA1002923 | Active | ||||||
14. | ALA224754 | 14 | Activity | 0 | ALA1002922 | Active | ||||||
15. | ALA224754 | 14 | Activity | 0 | ALA1002921 | Active | ||||||
16. | ALA224754 | 14 | Activity | 0 | ALA1002920 | Active | ||||||
17. | ALA224754 | 14 | EC50 | = | 10.8 | uM | ALA1002917 | 4.97 | nM | |||
18. | ALA224754 | 14 | EC50 | = | 12 | uM | ALA1002916 | 4.92 | nM | |||
19. | ALA224754 | 14 | Selectivity index | = | 4.2 | ALA918790 | ||||||
20. | ALA224754 | 14 | IC50 | = | 0.03 | uM | ALA918789 | 7.52 | nM | Homo sapiens |