# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA226880 | 1 | Activity | 0 | ALA2434593 | Dose-dependent effect | ||||||
2. | ALA226880 | 1 | Activity | 0 | ALA2434591 | Active | ||||||
3. | ALA226880 | 1 | Cp | = | 83 | nM | ALA2434589 | nM | Mus musculus | |||
4. | ALA226880 | 1 | Cp | = | 77 | nM | ALA2434586 | nM | Mus musculus | |||
5. | ALA226880 | 1 | Drug uptake | = | 412 | nM | ALA2434584 | nM | Mus musculus | |||
6. | ALA226880 | 1 | Drug uptake | = | 383 | nM | ALA2434585 | nM | Mus musculus | |||
7. | ALA226880 | 1 | AUC | = | 6245 | nM.hr | ALA2434583 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
8. | ALA226880 | 1 | AUC | = | 5536 | nM.hr | ALA2434588 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
9. | ALA226880 | 1 | Fu | = | 0.9 | % | ALA2434590 | Mus musculus | ||||
10. | ALA226880 | 1 | Fu | = | 0.5 | % | ALA2434582 | |||||
11. | ALA226880 | 1 | Activity | 0 | ALA2434581 | Active | Mus musculus | |||||
12. | ALA226880 | 1 | IC50 | = | 6.6 | nM | ALA962343 | 8.18 | nM | Homo sapiens | ||
13. | ALA226880 | 1 | IC50 | = | 4.2 | nM | ALA962342 | 8.38 | nM | Homo sapiens | ||
14. | ALA226880 | 1 | IC50 | = | 2.2 | nM | ALA962341 | 8.66 | nM | Homo sapiens | ||
15. | ALA226880 | 1 | IC50 | = | 6.2 | nM | ALA962340 | 8.21 | nM | Homo sapiens | ||
16. | ALA226880 | 1 | Activity | = | 82 | % | ALA965750 | % | Homo sapiens | |||
17. | ALA226880 | 1 | Activity | = | 14 | % | ALA965749 | % | Homo sapiens | |||
18. | ALA226880 | 1 | Activity | = | 4.2 | % | ALA965748 | % | Homo sapiens | |||
19. | ALA226880 | 1 | IC50 | = | 6.6 | nM | ALA965747 | 8.18 | nM | |||
20. | ALA226880 | 1 | IC50 | = | 4.2 | nM | ALA965746 | 8.38 | nM | Homo sapiens |