# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | UK 383367 | 1 | inhibition | = | -0.04 | % | ALA4513082 | % | Severe acute respiratory syndrome coronavirus 2 | |||
2. | UK 383367 | 1 | Inhibition | = | -1.507 | % | ALA4495582 | % | Severe acute respiratory syndrome coronavirus 2 | |||
3. | UK 383367 | 1 | inhibition | = | -0.04 | % | ALA4513082 | % | Severe acute respiratory syndrome coronavirus 2 | |||
4. | UK 383367 | 1 | inhibition | = | 23.54 | % | ALA4808150 | % | Homo sapiens | |||
5. | UK 383367 | 1 | inhibition | = | 24.04 | % | ALA4808149 | % | Homo sapiens | |||
6. | UK 383367 | 1 | Inhibition | = | 7.81 | % | ALA4303805 | % | Severe acute respiratory syndrome coronavirus 2 | |||
7. | UK 383367 | 1 | Potency | 0.008 | uM | ALA3215001 | inactive | nM | ||||
8. | UK 383367 | 1 | Potency | 16.774 | uM | ALA3214945 | inactive | nM | ||||
9. | UK 383367 | 1 | Potency | 21.118 | uM | ALA3214842 | inactive | nM | ||||
10. | UK 383367 | 1 | Potency | 21.118 | uM | ALA3214813 | inactive | nM | ||||
11. | UK 383367 | 1 | pKa | = | 9 | ALA941548 | ||||||
12. | UK 383367 | 1 | logD | = | 2.6 | ALA941547 | ||||||
13. | UK 383367 | 1 | IC50 | = | 0.9 | uM | ALA946663 | 6.05 | nM | Homo sapiens | ||
14. | UK 383367 | 1 | IC50 | = | 2.4 | uM | ALA946662 | 5.62 | nM | Homo sapiens | ||
15. | UK 383367 | 1 | IC50 | = | 1.5 | uM | ALA946661 | 5.82 | nM | Homo sapiens | ||
16. | UK 383367 | 1 | IC50 | = | 1.8 | uM | ALA946660 | 5.75 | nM | Homo sapiens | ||
17. | UK 383367 | 1 | INH | = | 69 | % | ALA946659 | % | ||||
18. | UK 383367 | 1 | solubility | = | 670 | ug ml-1 | ALA946658 | ug.mL-1 | ||||
19. | UK 383367 | 1 | TED | = | 1.59 | microg/cm2/h | ALA946657 | microg/cm2/h | Homo sapiens | |||
20. | UK 383367 | 1 | solubility | = | 13800 | ug ml-1 | ALA946656 | ug.mL-1 |