# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA396778 | (S)-7 | IC50 | = | 25.8 | nM | ALA2382556 | 7.59 | nM | Rattus norvegicus | ||
2. | ALA396778 | (S)-7 | Ratio IC50 | = | 1.4 | ALA2382554 | ||||||
3. | ALA396778 | (S)-7 | INH | 0 | ALA2382553 | Active | % | Homo sapiens | ||||
4. | ALA396778 | (S)-7 | IC50 | = | 7.67 | nM | ALA2382555 | 8.12 | nM | Homo sapiens | ||
5. | ALA396778 | (S)-7 | IC50 | = | 0.048 | uM | ALA4054025 | 7.32 | nM | Homo sapiens | ||
6. | ALA396778 | (S)-7 | IC50 | = | 100 | nM | ALA3706349 | 7.00 | 304399 | nM | Rattus norvegicus | |
7. | ALA396778 | (S)-7 | deltaTm | = | 6.6 | degrees C | ALA3404823 | degrees C | Homo sapiens | |||
8. | ALA396778 | (S)-7 | Ki | = | 16.7 | nM | ALA3407043 | 7.78 | nM | Homo sapiens | ||
9. | ALA396778 | (S)-7 | Ki | = | 5.4 | nM | ALA3404812 | 8.27 | nM | Homo sapiens | ||
10. | ALA396778 | (S)-7 | Activity | = | 31 | % | ALA3404819 | % | Rattus norvegicus | |||
11. | ALA396778 | (S)-7 | Activity | = | 100 | % | ALA3404820 | % | Rattus norvegicus | |||
12. | ALA396778 | (S)-7 | Kd | = | 187.2 | nM | ALA3404821 | 6.73 | nM | Homo sapiens | ||
13. | ALA396778 | (S)-7 | EC50 | = | 15 | uM | ALA3404822 | 4.82 | nM | Homo sapiens | ||
14. | ALA396778 | (S)-7 | IC50 | = | 5.18 | nM | ALA3364094 | 8.29 | nM | Homo sapiens | ||
15. | ALA396778 | (S)-7 | IC50 | = | 18 | nM | ALA3364095 | 7.75 | nM | Rattus norvegicus | ||
16. | ALA396778 | (S)-7 | Ratio IC50 | = | 5000 | ALA3364096 | ||||||
17. | ALA396778 | (S)-7 | Ratio IC50 | = | 23 | ALA3364099 | Homo sapiens | |||||
18. | ALA396778 | (S)-7 | IC50 | = | 45000 | nM | ALA3364088 | 4.35 | nM | Homo sapiens | ||
19. | ALA396778 | (S)-7 | IC50 | = | 580000 | nM | ALA3364089 | nM | Rattus norvegicus | |||
20. | ALA396778 | (S)-7 | IC50 | = | 9 | nM | ALA3364090 | 8.05 | nM | Homo sapiens |