| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA281724 | 54 | pKa | = | 2.85 | ALA3804245 | ||||||
| 2. | ALA281724 | 54 | IC50 | = | 40 | uM | ALA3803981 | 4.40 | nM | |||
| 3. | ALA281724 | 54 | Kd | = | 2.9 | uM | ALA3803975 | 5.54 | nM | Bos taurus | ||
| 4. | ALA281724 | 54 | IC50 | = | 14 | uM | ALA2416953 | 4.85 | nM | Homo sapiens | ||
| 5. | ALA281724 | 54 | IC50 | = | 5.7 | uM | ALA2416952 | 5.24 | nM | Homo sapiens | ||
| 6. | ALA281724 | 54 | INH | = | 4.3 | % | ALA2416954 | % | Homo sapiens | |||
| 7. | ALA281724 | 54 | INH | = | 5.2 | % | ALA2416955 | % | Homo sapiens | |||
| 8. | ALA281724 | 54 | Vdss | = | 2.6 | L/Kg | ALA1027763 | L.kg-1 | Homo sapiens | |||
| 9. | ALA281724 | 54 | t1/2 | = | 19.8 | hr | ALA1028547 | hr | Homo sapiens | |||
| 10. | ALA281724 | 54 | MRT | = | 23.3 | hr | ALA1028546 | hr | Homo sapiens | |||
| 11. | ALA281724 | 54 | CL | = | 1.54 | ml/min.kg | ALA1028545 | mL.min-1.kg-1 | Homo sapiens | |||
| 12. | ALA281724 | 54 | Vdss | = | 2.15 | L/Kg | ALA1028544 | L.kg-1 | Homo sapiens | |||
| 13. | ALA281724 | 54 | t1/2 | = | 23.5 | hr | ALA1028543 | hr | Homo sapiens | |||
| 14. | ALA281724 | 54 | MRT | = | 28.7 | hr | ALA1028542 | hr | Homo sapiens | |||
| 15. | ALA281724 | 54 | CL | = | 1.8 | ml/min.kg | ALA1028541 | mL.min-1.kg-1 | Homo sapiens | |||
| 16. | ALA281724 | 54 | Vdss | = | 3.1 | L/Kg | ALA1028540 | L.kg-1 | Homo sapiens | |||
| 17. | ALA281724 | 54 | Inhibition | = | 66 | % | ALA720015 | % | Mus musculus | |||
| 18. | ALA281724 | 54 | IC50 | = | 0.26 | uM | ALA806327 | 6.58 | nM | Rattus norvegicus | ||
| 19. | ALA281724 | 54 | Inhibition | 0 | ALA787012 | No data | % | Rattus norvegicus | ||||
| 20. | ALA281724 | 54 | IC50 | = | 2939 | nmol/l | ALA780515 | 5.53 | nM | Rattus norvegicus |
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