# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA393979 | 8b | Activity | = | 170.5 | g | ALA902780 | g | Rattus norvegicus | |||
2. | ALA393979 | 8b | Activity | = | 163.5 | g | ALA902779 | g | Rattus norvegicus | |||
3. | ALA393979 | 8b | IC50 | = | 4.5 | uM | ALA901754 | 5.35 | nM | Mus musculus | ||
4. | ALA393979 | 8b | IC50 | = | 45 | uM | ALA901753 | 4.35 | nM | Rattus norvegicus | ||
5. | ALA393979 | 8b | IC50 | = | 2.2 | uM | ALA901752 | 5.66 | nM | Rattus norvegicus | ||
6. | ALA393979 | 8b | IC50 | = | 4.8 | uM | ALA901751 | 5.32 | nM | Mus musculus | ||
7. | ALA393979 | 8b | IC50 | = | 0.008 | uM | ALA901750 | 8.10 | nM | Mus musculus | ||
8. | ALA393979 | 8b | IC50 | = | 0.025 | uM | ALA901749 | 7.61 | nM | Rattus norvegicus | ||
9. | ALA393979 | 8b | Stability | = | 81 | % | ALA901748 | % | Rattus norvegicus | |||
10. | ALA393979 | 8b | t1/2 | = | 3 | hr | ALA902761 | hr | ||||
11. | ALA393979 | 8b | t1/2 | = | 64 | hr | ALA902760 | hr | ||||
12. | ALA393979 | 8b | t1/2 | > | 2 | weeks | ALA902759 | hr | ||||
13. | ALA393979 | 8b | t1/2 | = | 35 | hr | ALA902758 | hr | ||||
14. | ALA393979 | 8b | Solubility | > | 200 | uM | ALA902757 | nM | ||||
15. | ALA393979 | 8b | Log D | = | -0.08 | ALA902756 | ||||||
16. | ALA393979 | 8b | Ratio IC50 | = | 9000 | ALA902795 | ||||||
17. | ALA393979 | 8b | Ratio IC50 | = | 300 | ALA902794 | ||||||
18. | ALA393979 | 8b | Ratio IC50 | = | 800 | ALA902742 | ||||||
19. | ALA393979 | 8b | Activity | = | 5 | % | ALA902793 | % | Rattus norvegicus | |||
20. | ALA393979 | 8b | Activity | = | 3 | % | ALA902787 | % | Rattus norvegicus |