| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA246356 | 5 | IC50 | = | 194 | nM | ALA887103 | 6.71 | nM | Homo sapiens | ||
| 2. | ALA246356 | 5 | Ratio IC50 | = | 63 | ALA887102 | Homo sapiens | |||||
| 3. | ALA246356 | 5 | Solubility | = | 0.003 | mg/ml | ALA887100 | ug.mL-1 | ||||
| 4. | ALA246356 | 5 | Solubility | = | 0.021 | mg/ml | ALA887099 | ug.mL-1 | ||||
| 5. | ALA246356 | 5 | MRT | = | 1.5 | hr | ALA887081 | hr | Rattus norvegicus | |||
| 6. | ALA246356 | 5 | t1/2 | = | 1.7 | hr | ALA887080 | hr | Rattus norvegicus | |||
| 7. | ALA246356 | 5 | AUC | = | 509 | ng.hr/ml | ALA887098 | ng.hr.mL-1 | Rattus norvegicus | |||
| 8. | ALA246356 | 5 | Cmax | = | 119 | ng/ml | ALA887097 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 9. | ALA246356 | 5 | F | = | 4 | % | ALA887096 | % | Rattus norvegicus | |||
| 10. | ALA246356 | 5 | IC50 | = | 40000 | nM | ALA887094 | 4.40 | nM | Homo sapiens | ||
| 11. | ALA246356 | 5 | Vdss | = | 1311 | ml/kg | ALA887095 | L.kg-1 | Rattus norvegicus | |||
| 12. | ALA246356 | 5 | IC50 | = | 25000 | nM | ALA887093 | 4.60 | nM | Homo sapiens | ||
| 13. | ALA246356 | 5 | IC50 | = | 25000 | nM | ALA887092 | 4.60 | nM | Homo sapiens | ||
| 14. | ALA246356 | 5 | IC50 | = | 25000 | nM | ALA887091 | 4.60 | nM | Homo sapiens | ||
| 15. | ALA246356 | 5 | IC50 | = | 25000 | nM | ALA887090 | 4.60 | nM | Homo sapiens | ||
| 16. | ALA246356 | 5 | IC50 | = | 25000 | nM | ALA887089 | 4.60 | nM | Homo sapiens | ||
| 17. | ALA246356 | 5 | IC50 | = | 17800 | nM | ALA887088 | 4.75 | nM | Homo sapiens | ||
| 18. | ALA246356 | 5 | IC50 | = | 5360 | nM | ALA887087 | 5.27 | nM | Homo sapiens | ||
| 19. | ALA246356 | 5 | IC50 | = | 2195 | nM | ALA887086 | 5.66 | nM | Homo sapiens | ||
| 20. | ALA246356 | 5 | IC50 | = | 1746 | nM | ALA887085 | 5.76 | nM | Homo sapiens |
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